Experimental methods in the study of thermodynamic polymorph stability relationships

American Pharmaceutical Review

Volumn 9, Issue 1, 2006, Pages 88-93

  Carlton, Robert A ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

BENZYL THIOCYANATE; SODIUM CHLORIDE;

ARTICLE; CALORIMETER; CRYSTALLOGRAPHY; DENSITY; ENANTIOTROPY; ENERGY; ENTHALPY; EXPERIMENTAL STUDY; GENETIC POLYMORPHISM; HEAT TRANSFER; MELTING POINT; MICROSCOPY; MONOTROPY; SOLID STATE; SOLUBILITY; TEMPERATURE; THERMODYNAMICS; VAPOR PRESSURE;

EID: 55549084893     PISSN: 10998012     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (13)

1. Bettinetti, G. (1988) Analysis of the Polymorphism of Drugs, Il Farmaco 43, 3 pp. 71-99.
2. Brittain, H.G. (1999) Polymorphism in Pharmaceutical Solids, Marcel Dekkar, New York.
3. Burger, A. (1982) Thermodynamic and other Aspects of the Polymorphism of Drugs, Pharmacy International, May, pp. 158-163.
4. Burger, A., Ramberger, R. (1979) Polymorphism of Pharmaceuticals and other Molecular Crystals. I. Theory of Thermodynamic Rules, Mikrochim. Acta, 2 pp 259-271.
5. Burger, A., Ramberger, R. (1979) Polymorphism of Pharmaceuticals and other Molecular Crystals. II. Applicability of Thermodynamic Rules, Mikrochim. Acta, 2 pp 273-316.
6. Haleblian, J., McCrone, W. (1969) Pharmaceutical Applications of Polymorphism, J of Pharm Sci, 58, 8 pp. 911-929.
7. Giron, D. (1995) Thermal Analysis and Calorimetric Methods in the Characterization of Polymorphs and Solvates, Thermochimica Acta, 248 pp. 1-59.
8. Grunenberg, J., Henck, O., Siesler, H.W. (1996) Theortical Derivation and Practical Application of Energy/Temperature Diagrams as an Instrument in Preformulation Studies of Polymorphic Drug Substances, International Journal of Pharmaceutics, 129 pp. 147-158.
9. Rodriquez-Spong, B., Price, C.P., Jayasankar, A., Matzger, A.J., Rodriguez-Hornedo, N. (2004) General Principles of Pharmaceutical Solid Polymorphism: a Supramolecular Perspective, Advanced Drug Delivery Reviews, 56 pp. 241-274.
10. Teetsov, A.S., McCrone, W.C. (1965) The Microscopical Study of Polymorph Stability Diagrams, The Microscope and Crystal Front, vol 5 no 1, pp 13-29.
11. Yu, L., Reutzel, S.M., Stephenson, G.A. (1998) Physical Characterization of Polymorphic Drugs: an Integrated Characterization Strategy, Pharm. Sci. Technol. Today, I pp 118-127.
12. Yu, L., Stephenson, G.A., Mitchell, C.A., Bunnell, C.A., Snorek, S.V., Bowyer, J.J., Borchardt, T.B., Stowell, J.G., Byrn, S.R. (2000) Thermochemistry and Conformational Polymorphism of a Hexamorphic Crystal System, J Am Chem Soc, 122, pp. 585-591.
13. Yu, L. (1995) Inferring Thermodynamic Stability Relationship from Melting Data, J. Pharm. Sci. pp 966-974.