Consequences of cis-amide bond simulation in opioid peptides

International Journal of Peptide Research and Therapeutics

Volumn 5, Issue 5-6, 1998, Pages 437-440

  Olczak, Jacek ^a   Kaczmarek, Krzysztof ^a   Maszczyńska, Iwona ^b   Lisowski, Marek ^c   Stropova, Dagmar ^d   Hruby, Victor J ^e   Yamamura, Henry I ^d   Lipkowski, Andrzej W ^b   Zabrocki, Janusz ^a  

^a LODZ UNIVERSITY OF TECHNOLOGY   (Poland)

^b MOSSAKOWSKI MEDICAL RESEARCH CENTRE   (Poland)

^c UNIVERSITY OF WROC AW   (Poland)

^d UNIVERSITY OF ARIZONA COLLEGE OF MEDICINE   (United States)

^e University of Arizona   (United States)

Author keywords

1,5 disubstituted tetrazole ring; Cis peptide bond conformation; Leu enkephalin

Indexed keywords

EID: 54749141627     PISSN: 15733149     EISSN: 15733904     Source Type: Journal    
DOI: 10.1007/BF02443502     Document Type: Article

References (5)

1. DiMaio, J., Nguen, T.M.-D., Lemieux, C. and Shiller, P.W., J. Med. Chem., 25 (1982) 1432.
2. Mosberg, H.I., Hurst, R., Hruby, V.J., Gee, K., Yamamura, H.I., Galligan, J.J. and Burks, T.F., Proc. Natl. Acad. Sci. USA, 80 (1983) 5871.
3. Belton, P., Cotton, R., Giles, M.B., Gormley, J.J., Miller, L., Shaw, J.S., Timms, D. and Wilkinson, A., Life Sci., 33 (Suppl. 1) (1983) 443.
4. Marshall, G.R., Humblet, C., Van Opdenbosch, N. and Zabrocki, J., In Rich, D.H. and Gross, E. (Eds.) Peptides: Synthesis-Structure-Function, (Proceedings of the 7th American peptide Symposium), Pierce Chemical Co., Rockford, IL, U.S.A., 1981, p. 669.
5. Zabrocki, J., Smith, G.D., Dunbar, J., Jijima, H. and Marshall, G.R., J. Am. Chem. Soc., 110 (1988) 5875.