Synthesis of RGD amphiphilic cyclic peptide as fibrinogen or fibronectin antagonist

International Journal of Peptide Research and Therapeutics

Volumn 4, Issue 4-6, 1997, Pages 455-461

  Sow, Mamadou Amadou ^a   Molla, Annie ^b   Lamaty, Frédéric ^a   Lazaro, René ^a  

^a UNIVERSITÉ DE MONTPELLIER   (France)

^b INSTITUT ALBERT BONNIOT   (France)

Author keywords

Aggregometry; Cyclic peptide; Diazaethyleneglycol derivative; HEL cell adhesion; RGD peptide

Indexed keywords

EID: 53249147858     PISSN: 15733149     EISSN: 15733904     Source Type: Journal    
DOI: 10.1007/BF02442916     Document Type: Article

References (28)

1. Ruoslahti, E. and Pierschbacher, M.D., Science, 238 (1987) 491.
2. Hynes, R.O., Cell, 48 (1987) 549.
3. Gartner, T.K. and Bennett, J.S., J. Biol. Chem., 260 (1985) 11891.
4. Samanen, J., Ali, F., Romoff, T., Calvo, R., Sorenson, E., Vasko, J., Storer, B., Berry, D., Bennett, D., Strohsacker, M., Powers, D., Stadel, J. and Nichols, A., J. Med. Chem., 34 (1991) 3114.
5. Aumailley, M., Gurrath, M., Müller, G., Calvete, J., Timpl, R. and Kessler, H., FEBS Lett., 291 (1991) 50.
6. For a recent review see: Ojima, I., Chakravarty, S. and Dong, Q., Bioorg. Med. Chem., 3 (1995) 337.
7. Hutchinson, J.H., Cook, J.J., Brashear, K.M., Breslin, M.J., Glass, J.D., Gould, R.J., Halczenko, W., Holahan, M.A., Lynch, R.J., Sitko, G.R., Stranieri, M.T. and Hartman, G.D., J. Med. Chem., 39 (1996) 4583.
8. Zablocki, J.A., Rico, J.G., Garland, R.B., Rogers, T.E., Williams, K., Schretzman, L.A., Rao, S.A., Bovy, P.R., Tjoeng, F.S., Lindmark, R.J., Toth, M.V., Zupec, M.E., McMackins, D.E., Adams, S.P., Miyano, M., Markos, C.S., Milton, M.N., Paulson, S., Herin, M., Jacqmin, P., Nicholson, N.S., Panzer-Knoddle, S.G., Haas, N.F., Page, J.D., Szalony, J.A., Taite, B.B., Salyers, A.K., King, L.W., Campion, J.G. and Feigen, L.P., J. Med. Chem., 38 (1995) 2378.
9. Hauzler, R., Gratias, R., Diefenbach, B., Goodman, S.L., Jonczyk, A. and Kessler, H., J. Am. Chem. Soc., 118 (1996) 7461.
10. Bach II, A.C., Espina, R., Jackson, S.A., Stouten, P.F.W., Duke, J.L., Mousa, S.A. and DeGrado, W.F., J. Am. Chem. Soc., 118 (1996) 293.
11. Nucci, M.L., Schorr, R. and Abuchowski, A., Adv. Drug Delivery Rev., 6 (1991) 133.
12. Kawasaki, K., Namikawa, M., Yamashiro, Y., Iwai, Y., Hama, T., Tsutsumi, Y., Yamamoto, S., Nakagawa, S. and Mayumi, T., Chem. Pharm. Bull., 43 (1995) 2133.
13. Cecchi, R., Rusconi, L., Tanzi, M.C. and Danusso, F., J. Med. Chem., 24 (1981) 622.
14. Zucker, M., Methods Enzymol., 169 (1988) 117.
15. Austel, V., Eisert, W.G., Himmelsbach, F., Linz, G., Muller, T.H., Pieper, H., Seewaldt-Becker, E. and Weisenberger, H., 207th American Chemical Society Meeting, Abstract MEDI 101, 28 March-2 April 1993.
16. Martin, P. and Papayamopoulo, I., Science, 216 (1982) 1233.
17. Lam, S.C.-T., Flow, E.F., Smith, M.A., Andneux, A., Ryckwaert, J.-J., Marguerie, G. and Ginsberg, M.H., J. Biol. Chem., 262 (1987) 947.
18. Kumagai, H., Tajima, M., Ueno, Y., Giga-Hama, Y. and Ohba, M., Biochem. Biophys. Res. Commun., 177 (1991) 74.
19. Bogusky, M.J., Naylor, A.M., Pitzenberger, S.M., Nutt, R.F., Brady, S.F., Colton, C.D., Sisko, J.T., Anderson, P.S. and Veber, D.F., Int. J. Pept. Protein Res., 39 (1992) 63.
20. Barker, P.L., Bullens, S., Bunting, S., Burdick, D.J., Chan, K.S., Deisher, T., Eigenbrot, C., Gadek, T.R., Gantzos, R., Lipari, M.T., Muir, C.D., Napier, M.A., Pitti, R.M., Padua, A., Quan, C., Stanley, M., Strable, M., Tom, J.Y.K. and Burnier, J.P., J. Med. Chem., 35 (1992) 2040.
21. Lender, A., Yao, W., Sprengeler, P.A., Spanevello, R.A., Furst, G.T., Hirschmann, R. and Smith III, A.B., Int. J. Pept. Protein Res., 42 (1993) 509.
22. Cheng, S., Craig, W.S., Mullen, D., Tschopp, J.F., Dixon, D. and Pierschbacher, M.D., J. Med. Chem., 37 (1994) 1.
23. Jackson, S., DeGrado, W., Dwivedi, A., Parthasarathy, A., Higley, A., Krywko, J., Rockwell, A., Markwalder, J., Wells, G., Wexler, R., Mousa, S. and Harlow, R., J. Am. Chem. Soc., 116 (1994) 3220.
24. Peishoff, C.E., Ali, F.E., Bean, J.W., Calvo, R., D'Ambrosio, C.A., Eggleston, D.S., Hwang, S.M., Kline, T.P., Koster, P.F., Nichols, A., Powers, D., Romoff, T., Samanen, J.M., Stadel, J., Vasko, J.A. and Kopple, K.D., J. Med. Chem., 35 (1992) 3962.
25. Cook, R.M., Adams, J.H. and Hudson, J.H., Tetrahedron Lett., 35 (1994) 6777.
26. Mitsunobu, O., Synthesis, (1981) 1.
27. Jouin, P., Poncet, J., Dufour, M.-N., Pantaloni, A. and Castro, B., J. Org. Chem., 54 (1989) 617.
28. Rodriguez, M., Amblard, M., Calas, M.C., Lignon, M.-F. and Martinez, J., Int. J. Pept. Protein Res., 35 (1990) 441.