AROMATIZATION;
ARTICLE;
CARBON NUCLEAR MAGNETIC RESONANCE;
CHEMICAL REACTION;
DRUG STRUCTURE;
DRUG SYNTHESIS;
INFRARED SPECTROSCOPY;
ONE POT SYNTHESIS;
POLYMERIZATION;
PROTON NUCLEAR MAGNETIC RESONANCE;
ROOM TEMPERATURE;
Benzo[b]thiophene as a template for substituted quinolines and tetrahydroquinolines
Chabert, J. F. D.; Rostaing, S. P.; Bouchu, D.; Lemaire, M. Benzo[b]thiophene as a template for substituted quinolines and tetrahydroquinolines. Tetrahedron Lett. 2006, 47, 1015-1018.
Discovery of novel quinoline-based estrogen receptor ligands using peptide interaction profiling
Hoekstra, W. J.; Patel, H. S.; Liang, X.; Blanc, J. B. E.; Heyer, D. O.; Wilson, T. M.; Iannone, M. A.; Kadwell, S. H.; Miller, L. A.; Pearce, K. H.; Simmons, C. A.; Shearin, J. Discovery of novel quinoline-based estrogen receptor ligands using peptide interaction profiling. J. Med. Chem. 2005, 48, 2243-2247;
A new series of PDGF receptor tyrosine kinase inhibitors: 3-substituted quinoline derivatives
(b) Maguire, M. P.; Sheets, K. R.; McVety, K.; Spada, A. P.; Zilberstein, A. A new series of PDGF receptor tyrosine kinase inhibitors: 3-substituted quinoline derivatives. J. Med. Chem. 1994, 37, 2129-2137.
Martinelline and martinellic acid, novel G-protein linked receptor antagonists from the tropical plant martinella iquitosensis (bignoniaceae)
Witherup, K. M.; Ransom, R. W.; Graham, A. C.; Bernard, A. M.; Salvatore, M. J.; Lumma, W. C.; Anderson, P. S.; Pitzerberger, S. M.; Varga, S. L. Martinelline and martinellic acid, novel G-protein linked receptor antagonists from the tropical plant martinella iquitosensis (bignoniaceae). J. Am. Chem. Soc. 1995, 117, 6682-6685;
Anticonvulsant activity of glycine-site NMDA antagonists. 2. trans 2-carboxy-4-substituted tetrahydroquinolines
(b) Carling, R. W.; Leeson, P. D.; Moseleyy, A. M.; Smith, J. D.; Saywell, K.; Tricklebank, M. D.; Kemp, J. A.; Marshall, G. R.; Foster, A. C.; Grimwood, S. Anticonvulsant activity of glycine-site NMDA antagonists. 2. trans 2-carboxy-4-substituted tetrahydroquinolines. Bioorg. Med. Chem. Lett. 1993, 3, 65-70.
A. R. Katritzky, C. W. Rees, E. F. V. Scriven Eds, Pergamon Press: Oxford
(b) Balasubramanian, M.; Keay, J. G. In Comprehensive Heterocyclic Chemistry II, A. R. Katritzky, C. W. Rees, E. F. V. Scriven (Eds.), Pergamon Press: Oxford, 1996; vol. 5, pp. 245-265;
Synthesis and antibacterial evaluation of certain quinolone derivatives
(c) Chen, Y. L.; Fang, K. C.; Sheu, J. Y.; Hsu, S. L.; Tzeng, C. C. Synthesis and antibacterial evaluation of certain quinolone derivatives. J. Med. Chem. 2001, 44, 2374-2377;
Roma, G.; Braccio, M. D.; Grossi, G.; Mattioli, F.; Ghia, M. 1,8-naphthyridines IV. 9-substituted N,N-dialkyl-5-(alkylamino or cycloalkylamino) [1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides, new compounds with anti-aggressive and potent anti-inflammatory activities. Eur. J. Med. Chem. 2000, 35, 1021-1035;
(d) Roma, G.; Braccio, M. D.; Grossi, G.; Mattioli, F.; Ghia, M. 1,8-naphthyridines IV. 9-substituted N,N-dialkyl-5-(alkylamino or cycloalkylamino) [1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides, new compounds with anti-aggressive and potent anti-inflammatory activities. Eur. J. Med. Chem. 2000, 35, 1021-1035;
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Total synthesis of (±)-virantmycin and determination of its stereochemistry
(e) Morimoto, Y.; Matsuda, F.; Shirahama, H. Total synthesis of (±)-virantmycin and determination of its stereochemistry. Synlett. 1991, 202-203;
Potential antitumor agents. 57. 2-phenylquinoline-8-carboxamides as "minimal" DNA-intercalating antitumor agents with in vivo solid tumor activity
Atwell, G. J.; Baguley, B. C.; Denny, W. A. Potential antitumor agents. 57. 2-phenylquinoline-8-carboxamides as "minimal" DNA-intercalating antitumor agents with in vivo solid tumor activity. Med. Chem. 1989, 32, 396-401.
Synthesis and characterization of quinoline derivatives via the Friedländer reaction
Yang, D.; Jiang, K.; Li, J.; Xu, F. Synthesis and characterization of quinoline derivatives via the Friedländer reaction. Tetrahedron 2007, 63, 7654-7658.
Recent advances in the biginelli dihydropyrimidine synthesis. New tricks from an old dog
For a more recent update on the Biginelli reaction, see
For a more recent update on the Biginelli reaction, see: Kappe, C. O. Recent advances in the biginelli dihydropyrimidine synthesis. New tricks from an old dog. Acc. Chem. Res. 2000, 33, 879-888.
Molecular iodine-catalyzed one-pot synthesis of substituted quinolines from imines and aldehydes
Lin, X. F.; Cui, S. L.; Wang, Y. G. Molecular iodine-catalyzed one-pot synthesis of substituted quinolines from imines and aldehydes. Tetrahedron Letters 2006, 47, 3127-3130.
