Design and study of rifampicin oral controlled release formulations

Drug Delivery: Journal of Delivery and Targeting of Therapeutic Agents

Volumn 11, Issue 5, 2004, Pages 311-317

  Hiremath, S P ^a   Saha, R N ^a  

^a BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

Controlled Release; Hydroxypropyl Methylcellulose; Rifampicin; Zero Order

Indexed keywords

EXCIPIENT; HYDROXYPROPYLMETHYLCELLULOSE; POLYMER; RIFAMPICIN;

ARTICLE; COMPRESSION; CONTROLLED DRUG RELEASE; CONTROLLED RELEASE FORMULATION; DRUG STABILITY; DRUG STORAGE; FORCE; KINETICS; MATHEMATICAL ANALYSIS; PRIORITY JOURNAL; RITGER PEPPAS EXPONENTIAL EQUATION; TABLET FORMULATION; TABLET PROPERTY;

ALGORITHMS; ANTIBIOTICS, ANTITUBERCULAR; CHEMISTRY, PHARMACEUTICAL; COMPRESSIVE STRENGTH; DELAYED-ACTION PREPARATIONS; DRUG STABILITY; METHYLCELLULOSE; REPRODUCIBILITY OF RESULTS; RIFAMPIN; SOLUBILITY; TABLETS;

EID: 4944247160     PISSN: 10717544     EISSN: None     Source Type: Journal    
DOI: 10.1080/10717540490494087     Document Type: Article

References (21)

1. Colombo, P. 1993. Swelling-controlled release in hydrogel matrices for oral route. Adv. Drug Del. Rev. 11:37-57.
2. Hara, P. O., and Hickey, A. J. 2000. Respirable PLGA microspheres containing rifampicin for the treatment of tuberculosis: manufacture and characterization. Pharm. Res. 17(8):955-961.
3. Indian Pharmacopoeia, vol II. 1996. Government of India Ministry of Health and Family Welfare. New Delhi: The Controller Publications, 665-666.
4. Khan, G. M., and Zhu, J.-B. 1999. Studies on drug release kinetics fro ibuprofen-carbomer hydrophilic matrix tablets: influence of co-excipients on release rate of the drug. J. Control. Rel. 57:197-203.
5. Kim, H., and Fassihi, R. 1997. Application of binary polymer system in drug release rate modulation. 2. Influence of formulation variables and hydrodynamic conditions on release kinetics. J. Pharm. Sci. 86(3):323-328.
6. Korsenmeyer, R. W., and Peppas, N. A. 1983. Macromolecular and modelling aspects of swelling-controlled systems. In Controlled Release Delivery Systems, eds. S. Z. Mansdorf and T. J. Roseman, 77. New York: Dekker.
7. Lee, B.-J., Ryu, S.-G., and Cui, J.-H. 1999. Formulation and release characteristics of hydroxypropyl methylcellulose matrix tablet containing melatonin. Drug Dev. Ind. Pharm. 25(4):493-501.
8. Narasimhan, B., and Peppas, N. A. 1996. Disentanglement and reptation during dissolution of rubbery polymers. J. Polym. Sci. Polym. Phys. 34:947-961.
9. Narasimhan, B., and Peppas, N. A. 1997. Molecular analysis of drug delivery systems controlled by dissolution of the polymer carrier. J. Pharm. Sci. 86:297-304.
10. Nokhodchi, A., Ford, J. L., Rowe, P. H., and Rubinstein, M. H. 1996. The effects of compression rate and force on the compaction properties of different viscosity grades of hydroxypropyl methylcellulose. Int. J. Pharm. 129:21-31.
11. Ranga Rao, K. V., Padmalatha Devi, K., and Buri, B. 1988. Cellulose matrices for zero-order release of soluble drugs. Drug Dev. Ind. Pharm. 14:2299-2320.
12. Rao, B. S., and Murthy, K. V. R. 2000. Preparation and in vitro evaluation of chitosan matrices cross-linked by formaldehyde vapors. Drug Dev. Ind. Pharm. 26(10):1085-1090.
13. Rao, B. S., and Murthy, K. V. R. 2001. Development of dissolution medium for rifampicin sustained release formulations. Ind. J. Pharm. Sci. 63(3):258-260.
14. Rao, B. S., and Murthy, K. V. R. 2002. Studies on rifampicin release from ethylcellulose coated nonpareil beads. Int. J. Pharm. 231:97-106.
15. Rao, S. B., Seshasayana, A., Narayan, C. P. S., Sudha, K. S., Saradhi, S. V. P., Ravi Kumar, N., and Murthy, K. V. R. 2001. Studies on release of rifampicin from sintered matrix tablets. Ind. J. Pharm. Sci. 63(5):371-378.
16. Ritger, P. L., and Peppas, N. A. 1987. A simple equation for description of solute release. II. Fickian and anomalous release from swellable devices. J. Control. Rel. 5:37-42.
17. Seshasayana, A., Rao, S. B., Raju, Y. P., Narayan, C. P. S., and Murthy, K. V. R. 2001. Studies on release of rifampicin from modified pulsnicap technique. Ind. J. Pharm. Sci. 63(4):337-339.
18. Varghas, C. I., and Ghaly, E. S. 1999. Kinetic release of theophyline from hydrophilic swellable matrices. Drug Dev. Ind. Pharm. 25(9):1045-1050.
19. Vazquez, M. J., Perez-Marcos, B., Gomez-Amoza, J. L., Martinez-Pacheco, R., Souto, C., and Concheiro, A. 1992. Influence of technological variables on release of drugs from hydrophilic matrices. Drug Dev. Ind. Pharm. 18:1355-1375.
20. Velasco, M., Ford, J. L., Rowe, P., and Rajabi-Siahboomi, A. R. 1999. Influence of drug: hydroxypropyl methylcellulose ratio, drug and polymer particle size and compression force on the release of diclofenac sodium from HPMC matrices. J. Control. Rel. 57:75-85.
21. York, P. 1979. A consideration of experimental variables in the analysis of powder scompaction behavior. J. Pharm. Pharmacol. 31:244-246.