Kinetic and thermodynamic analysis of 10-hydroxy-camptothecin hydrolysis at physiological pH

Journal of Chemical Thermodynamics

Volumn 40, Issue 9, 2008, Pages 1439-1444

  Kunadharaju, Sasank ^a   Savva, Michalakis ^a  

^a LONG ISLAND UNIVERSITY   (United States)

Author keywords

10 Hydroxy camptothecin; Derivative spectroscopy; Energy of activation; Frequency factor; Hydrolysis kinetics; Thermodynamics

Indexed keywords

BODY FLUIDS; CARBOXYLATION; HYDROLYSIS; PARAMETER ESTIMATION; PH EFFECTS; PHYSIOLOGICAL MODELS; RATE CONSTANTS; THERMOANALYSIS; THERMODYNAMICS;

10-HYDROXY-CAMPTOTHECIN; ANALYTICAL METHODS; CAMPTOTHECIN; DERIVATIVE SPECTROSCOPY; ENERGY OF ACTIVATION; FREQUENCY FACTOR; HYDROLYSIS KINETICS; LACTONE RINGS; PHYSIOLOGICAL PH; REPRODUCIBILITY; SIMULTANEOUS ESTIMATION; THERMODYNAMIC ANALYSIS;

PH;

EID: 49049089946     PISSN: 00219614     EISSN: 10963626     Source Type: Journal    
DOI: 10.1016/j.jct.2008.04.015     Document Type: Article

References (20)

1. Wall M.E., Wani M.C., Nicholas A.W., Manikumar G., Tele C., Moore L., Truesdale A., Leitner P., and Besterman J.M. J. Med. Chem. 36 (1993) 2689-2700
2. Gottlieb J.A., Guarino A.M., Call J.B., Oliverio V.T., and Block J.B. Cancer Chemother. Rep. 54 (1970) 461-470
3. Wani M.C., Ronman P.E., Lindley J.T., and Wall M.E. J. Med. Chem. 23 (1980) 554-560
4. Jaxel C., Kohn K.W., Wani M.C., Wall M.E., and Pommier Y. Cancer Res. 49 (1989) 1465-1469
5. Kingsbury W.D., Boehm J.C., Jakas D.R., Holden K.G., Hecht S.M., Gallagher G., Caranfa M.J., McCabe F.L., Faucette L.F., Johnson R.K., et al. J. Med. Chem. 34 (1991) 98-107
6. Kawato Y., Aonuma M., Hirota Y., Kuga H., and Sato K. Cancer Res. 51 (1991) 4187-4191
7. Kepler J.A., Wani M.C., McNaull J.N., Wall M.E., and Levine S.G. J. Org. Chem. 34 (1969) 3853-3858
8. Hsiang Y.H., Lihou M.G., and Liu L.F. Cancer Res. 49 (1989) 5077-5082
9. Hertzberg R.P., Caranfa M.J., and Hecht S.M. Biochemistry 28 (1989) 4629-4638
10. Bjornsti M.A., Benedetti P., Viglianti G.A., and Wang J.C. Cancer Res. 49 (1989) 6318-6323
11. Gottlieb J.A., and Luce J.K. Cancer Chemother. Rep. 56 (1972) 103-105
12. Moertel C.G., Schutt A.J., Reitemeier R.J., and Hahn R.G. Cancer Chemother. Rep. 56 (1972) 95-101
13. Burke T.G., Mishra A.K., Wani M.C., and Wall M.E. Biochemistry 32 (1993) 5352-5364
14. Burke T.G., and Mi Z. J. Med. Chem. 37 (1994) 40-46
15. Mi Z., and Burke T.G. Biochemistry 33 (1994) 10325-10336
16. B. Selvi, S. Patel, M. Savva, J. Pharm. Sci. (2008), inpress.
17. Fassberg J., and Stella V.J. J. Pharm. Sci. 81 (1992) 676-684
18. Klopas A., Panderi I., and Parissi-Poulou M. J. Pharm. Biomed. Anal. 17 (1998) 515-524
19. Morelli B. J. Pharm. Biomed. Anal. 13 (1995) 219-227
20. Chourpa I., Millot J.M., Sockalingum G.D., Riou J.F., and Manfait M. Biochim. Biophys. Acta 1379 (1998) 353-366