Structure-activity study of phosphoramido acid esters as acetylcholinesterasf inhibitors

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 23, Issue 4, 2008, Pages 556-561

  Ghadimi, Saied ^a   Ebrahimi Valmoozi, Ali Asghar ^a   Pourayoubi, Mehrdad ^a   Asad Samani, Keyvan ^a  

^a IMAM HOSSEIN UNIVERSITY   (Iran)

Author keywords

Acetylcholinesterase; IC50; Inhibition; Lipophilicity; Phosphoramido acid ester; Structure activity study; X ray crystallography

Indexed keywords

ACETYLCHOLINESTERASE; INSECTICIDE; PHOSPHORAMIDO ACID ESTER DERIVATIVE; PHOSPHORAMIDOUS ACID DERIVATIVE;

ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CHEMICAL STRUCTURE; CHOLINESTERASE INHIBITION; COMPUTER PROGRAM; CONTROLLED STUDY; INFRARED SPECTROSCOPY; LIPOPHILICITY; MASS SPECTROMETRY; PHOSPHORUS NUCLEAR MAGNETIC RESONANCE; PREDICTION; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ACETYLCHOLINESTERASE; CHOLINESTERASE INHIBITORS; CRYSTALLOGRAPHY, X-RAY; ESTERS; HUMANS; KINETICS; ORGANOPHOSPHORUS COMPOUNDS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 48549103947     PISSN: 14756366     EISSN: 14756374     Source Type: Journal    
DOI: 10.1080/14756360701731981     Document Type: Article

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