Fluorinated estradiol derivatives for oestrogen receptor imaging: Impact of substituents, formulation and specific activity on the biodistribution in breast tumour-bearing mice

European Journal of Nuclear Medicine and Molecular Imaging

Volumn 35, Issue 8, 2008, Pages 1473-1479

  Bénard, François ^a   Ahmed, Naseem ^a   Beauregard, Jean Mathieu ^a   Rousseau, Jacques ^a   Aliaga, Antonio ^a   Dubuc, Céléna ^a   Croteau, Etienne ^a   Van Lier, Johan E ^a  

^a UNIVERSITY OF SHERBROOKE   (Canada)

Author keywords

4 fluoroestradiol; 18F 16 fluoroestradiol; Breast cancer; Oestrogen receptors; Positron emission tomography

Indexed keywords

11BETA METHOXY 16ALPHA FLUOROESTRADIOL F18; 16ALPHA FLUOROESTRADIOL F18; 2 FLUORO 11BETA METHOXY 16ALPHA FLUOROESTRADIOL F18; 4 FLUORO 11BETA METHOXY 16ALPHA FLUOROESTRADIOL F18; 4 FLUORO 16ALPHA FLUOROESTRADIOL F18; ALCOHOL; ESTRADIOL DERIVATIVE; ESTROGEN RECEPTOR; LIPID EMULSION; RADIOPHARMACEUTICAL AGENT; SODIUM CHLORIDE; UNCLASSIFIED DRUG; 4 FLUOROESTRADIOL; 4-FLUOROESTRADIOL; DIAGNOSTIC AGENT; DRUG DERIVATIVE; ESTRADIOL;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; BREAST TUMOR; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DRUG DISTRIBUTION; DRUG FORMULATION; DRUG TISSUE LEVEL; DRUG UPTAKE; FEMALE; IMAGING; ISOTOPE LABELING; MOUSE; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; PROTEIN EXPRESSION; RADIOACTIVITY; RECEPTOR DENSITY; UTERUS; ANIMAL; ANTIBODY SPECIFICITY; BAGG ALBINO MOUSE; METABOLISM; SCINTISCANNING; TISSUE DISTRIBUTION;

ANIMALS; BREAST NEOPLASMS; ESTRADIOL; MICE; MICE, INBRED BALB C; ORGAN SPECIFICITY; RADIOPHARMACEUTICALS; RECEPTORS, ESTROGEN; TISSUE DISTRIBUTION;

EID: 48149114857     PISSN: 16197070     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00259-008-0745-x     Document Type: Article

References (23)

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