Synthesis and biological evaluation of a focused library of beauveriolides

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 15, 2008, Pages 4397-4400

  Nagai, Kenichiro ^a   Doi, Takayuki ^b   Ohshiro, Taichi ^a   Sunazuka, Toshiaki ^a   Tomoda, Hiroshi ^a   Takahashi, Takashi ^b   Omura, Satoshi ^a  

^a KITASATO UNIVERSITY   (Japan)

^b TOKYO INSTITUTE OF TECHNOLOGY   (Japan)

Author keywords

ACAT; Antiatherogenic activity; Cyclic depsipeptide; Focused library

Indexed keywords

3 HYDROXY 4 METHYLOCTANOIC ACID; ALANINE; BEAUVERIOLIDE 1; BEAUVERIOLIDE 3; DEPSIPEPTIDE; ISOLEUCINE; OCTANOIC ACID DERIVATIVE; PHENYLALANINE; UNCLASSIFIED DRUG;

ARTICLE; BIOLOGICAL ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; LIPID STORAGE; SOLUBILITY;

ALANINE; AMINO ACIDS; ANIMALS; ATHEROSCLEROSIS; COMBINATORIAL CHEMISTRY TECHNIQUES; DEPSIPEPTIDES; DISEASE MODELS, ANIMAL; ISOLEUCINE; LIPID METABOLISM; MACROPHAGES; MICE; MOLECULAR STRUCTURE; STEROL O-ACYLTRANSFERASE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 47749149909     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.06.054     Document Type: Article

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