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Volumn 2, Issue 4, 2007, Pages 479-487

Design, synthesis, and evaluation of tripeptidic promoieties targeting the intestinal peptide transporter hPEPT1

(7) Thorn, Karina a Andersen, Rikke a Christensen, Jon a Jakobsen, Palle b Nielsen, Carsten Uhd a Steffansen, Bente a Begtrup, Mikael a

a UNIVERSITY OF COPENHAGEN (Denmark)

b NOVO NORDISK A S (Denmark)

Author keywords

Binding affinity; hPEPT1; Promoiety; Solid phase synthesis; Translocation

Indexed keywords

COTRANSPORTER; PEPTIDE; PRODRUG; SLC15A1 PROTEIN, HUMAN; UNCLASSIFIED DRUG;

ARTICLE; CELL STRAIN CACO 2; CHEMISTRY; DRUG ANTAGONISM; DRUG DESIGN; HELA CELL; HUMAN; STRUCTURE ACTIVITY RELATION;

CACO-2 CELLS; DRUG DESIGN; HELA CELLS; HUMANS; PEPTIDES; PRODRUGS; STRUCTURE-ACTIVITY RELATIONSHIP; SYMPORTERS;

EID: 47549113101 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200600200 Document Type: Article

Times cited : (8)

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