Thermal and non-thermal methods to evaluate compatibility of granisetron hydrochloride with tablet excipients

Pharmazie

Volumn 63, Issue 6, 2008, Pages 453-458

  Late, S G ^a   Banga, A K ^a  

^a MERCER UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 HYDROXYPROPYL BETA CYCLODEXTRIN; BETA CYCLODEXTRIN; CROSCARMELLOSE SODIUM; CROSPOVIDONE; ETHYL CELLULOSE; EXCIPIENT; GLUCOSE; GRANISETRON; HYDROXYPROPYLMETHYLCELLULOSE; LACTOSE; MAGNESIUM STEARATE; MANNITOL; MICROCRYSTALLINE CELLULOSE; TALC;

ARTICLE; DIFFERENTIAL SCANNING CALORIMETRY; DRUG EXCIPIENT COMPATIBILITY; INFRARED SPECTROSCOPY; PHARMACEUTICS; TABLET; THIN LAYER CHROMATOGRAPHY;

ANTIEMETICS; BETA-CYCLODEXTRINS; CALORIMETRY, DIFFERENTIAL SCANNING; CHEMISTRY, PHARMACEUTICAL; CHROMATOGRAPHY, THIN LAYER; EXCIPIENTS; GLUCOSE; GRANISETRON; MANNITOL; METHYLCELLULOSE; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; TABLETS; TEMPERATURE;

EID: 46849120801     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: 10.1691/ph.2008.7405     Document Type: Article

References (24)

1. Araujo AAS, Storpiritis S, Mercuri LP, Carvalho FMS, Filho MS, Matos JR (2003) Thermal analysis of antiretroviral zidovudine (AZT) and evaluation of the compatibility with excipients used in solid dosage forms. Int J Pharm 260: 303-314.
2. Arias MJ, Gines J.M, Moyano JR, Perez-Martinez JI, Rabasco AM (1995) Influence of the preparation method of solid dispersions on their dissolution rate: study of triamterene-D-mannitol system. Int J Pharm 123: 25-31.
3. Boscolo M, Carli F, Crimella T, Filippis P, De Ponti R, Furiosi G, Maf-fione G, Pasini M, Scarpetti G (1990) Evaluation on the suitability of differential scanning calorimetry in the preformulation stability screening. Acta Tech Legis Med 1: 29-47.
4. Botha SA, Lotter AP (1989) Compatibility study between ketoprofen and tablet excipients using differential scanning calorimetry. Drug Dev Ind Pharm 15: 415-426.
5. Chaturvedula A, Joshi DP, Anderson C, Morris R, Sembrowich WL, Ban-ga AK (2005) Dermal, subdermal and systemic concentrations of grani-setron by iontophoretic delivery. Pharm Res 22: 1313-1319.
6. Corvi Mora P, Cirri M, Mura P (2006) Differential scanning calorimetry as a screening technique in compatibility studies of DHEA extended release formulations. J Pharm Biomed Anal 42: 3-10.
7. Ford JL (1993) The use of thermal analysis in preformulation compatibility testing. Acta of symposium on Pharmacy and Thermal Analysis, Freiburg, p. 2.
8. Gilani K, Najafabadi AR, Barghi M, Rafiee-Tehrani M (2004) Aerosolization of beclomethasone dipropionate using spray dried lactose polyethylene glycol carriers. Eur J Pharm Biopharm 58: 595-606.
9. Gu L, Strickley RG, Chi L, Chowhan ZT (1990) Drug-excipient incompatibility studies of the dipeptide angiotensin converting enzyme inhibitor, Moexipril hydrochloride: dry powder vs wet granulation. Pharm Res 7: 379-383.
10. Joshi BV, Patil VB, Pokharkar VB (2002) Compatibility studies between carbamazepine and tablet excipients using thermal and non-thermal methods. Drug Dev Ind Pharm 28: 687-694.
11. Lin SY, Han RY (1992) Differential Scanning calorimetry as a screening technique to determine the compatibility of salbutamol sulfate with excipients. Pharmazie 47: 266-268.
12. Malan CEP, De Villiers MM, Lotter AP (1997) Application of differential scanning calorimetry and high performance liquid chromatography to determine the effects of mixture composition and preparation during the evaluation of niclosamide-excipient compatibility. J Pharm Biomed Anal 15: 549-557.
13. Mura P, Manderioli A, Bramanti G, Furlanetto S, Pinzauti S (1995) Utilization of differential scanning calorimetry as a screening technique to determine the compatibility of ketoprofen with excipients. Int J Pharm 119: 71-79.
14. Mura P, Faucci MT, Manderioli A, Bramanti G, Ceccarelli J (1998) Compatibility study of ibuproxam and pharmaceutical excipients using differential scanning calorimetry, hot stage microscopy and scanning electron microscopy. J Pharm Biomed Anal 18: 151-163.
15. Nassab PR, Rajko R, Sazobe-Revesz, P (2006) Physicochemical characterization of meloxicam-mannitol binary systems. J Pharm Biomed Anal 41: 1991-1197.
16. Okonogi S, Oguchi T, Yonemochi E, Puttipipatkhachorn S, Yamamoto K (1997) Improved dissolution of ofloxacin via solid dispersion. Int J Pharm 156: 175-180.
17. Rawat S, Jain SK (2004) Solubility enhancement of celecoxib using β-cyclodextrin inclusion complexes. Eur J Pharm Biopharm 57: 263-267.
18. Serajuddin ATM, Thakur AB, Ghoshal RN, Fakes SA, Randive KR, Morris KR, Varia SA (1999) Selection of solid dosage form composition through drug-excipient compatibility testing. J Pharm Sci 88: 696-704.
19. Smith A (1982) Use of thermal analysis in predicting drug-excipient interactions. Anal Proc 19: 559-561.
20. Tomassetti M, Catalani A, Rossi V, Vecchio S (2005) Thermal analysis study of the interaction between acetaminophen and excipients in solid dosage forms and in some binary mixtures. J Pharm Biomed Anal 37: 949-955.
21. Van Dooren AA, Duphar BV (1983) Design of drug-excipient interaction studies. Drug Dev Ind Pharm 9: 43-55.
22. Verma RK, Garg S (2005) Selection of excipients for extended release formulation of glipizide through drug-excipient compatibility testing. J Pharm Biomed Anal 38: 633-644.
23. Ventura CA, Tommasini S, Falcone A, Giannone I, Paolino D, Sdrafkakis V, Mondello MR, Puglisi G (2006) Influence of modified cyclodextrins on solubility and percutaneous absorption of celecoxib through human skin. Int J Pharm 314: 37-45.
24. Watson ES, O'Neill MJ, Justin J, Brenner N (1964) A Differential Scanning Calorimeter for quantitative differential thermal analysis. Anal Chem 36: 1233-1238.