메뉴 건너뛰기




Volumn 122, Issue 2, 2004, Pages 139-146

Pharmacological and functional biochemical properties of D-Ala 2-D-Nle5-enkephalin-Arg-Phe

Author keywords

CHO cells; Enkephalins; G protein stimulation; Opioid receptor; Radioligand binding; Tail withdrawal

Indexed keywords

APROTININ; BACITRACIN; CYPRODIME; DELTA OPIATE RECEPTOR; ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE]; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); KAPPA OPIATE RECEPTOR; METENKEPHALIN DERIVATIVE; METENKEPHALIN[2 DEXTRO ALANINE 6 ARGININE 7 PHENYLALANINE]; METENKEPHALIN[6 ARGININE 7 PHENYLALANINE]; MU OPIATE RECEPTOR; MU OPIATE RECEPTOR ANTAGONIST; NALOXONE; NALTRINDOLE; NORBINALTORPHIMINE; TYROSYL DEXTRO ALANYLGLYCYLPHENYLALANYL DEXTRO NORLEUCYLARGINYLPHENYLALANINE; UNCLASSIFIED DRUG;

EID: 4544278750     PISSN: 01670115     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.regpep.2004.06.017     Document Type: Article
Times cited : (3)

References (43)
  • 1
    • 0018346407 scopus 로고
    • Nucleotide sequence of cloned cDNA for bovine corticotropin-beta- lipotropin precursor
    • Nakanishi S., Inoue A., Kita T., Nakamura M., Chang A.C.Y., Cohen S.N., et al. Nucleotide sequence of cloned cDNA for bovine corticotropin-beta- lipotropin precursor. Nature. 278:1979;423-427
    • (1979) Nature , vol.278 , pp. 423-427
    • Nakanishi, S.1    Inoue, A.2    Kita, T.3    Nakamura, M.4    Chang, A.C.Y.5    Cohen, S.N.6
  • 2
    • 0019977784 scopus 로고
    • Cloning and sequence analysis of cDNA for porcine beta-neoendorphin/ dynorphin precursor
    • Kakidani H., Furutani Y., Takahashi H., Noda M., Morimoto Y., Hirose T., et al. Cloning and sequence analysis of cDNA for porcine beta-neoendorphin/ dynorphin precursor. Nature. 298:1982;245-249
    • (1982) Nature , vol.298 , pp. 245-249
    • Kakidani, H.1    Furutani, Y.2    Takahashi, H.3    Noda, M.4    Morimoto, Y.5    Hirose, T.6
  • 3
    • 0020048094 scopus 로고
    • Cloning and sequence analysis of cDNA for bovine adrenal proenkephalin
    • Noda M., Furutani Y., Takahashi H., Toyosato M., Hirose T., Inayama S., et al. Cloning and sequence analysis of cDNA for bovine adrenal proenkephalin. Nature. 295:1982;202-206
    • (1982) Nature , vol.295 , pp. 202-206
    • Noda, M.1    Furutani, Y.2    Takahashi, H.3    Toyosato, M.4    Hirose, T.5    Inayama, S.6
  • 6
    • 0037680794 scopus 로고    scopus 로고
    • Characterization of zebrafish proenkephalin reveals novel opioid sequences
    • Gonzalez N.V., Gonzalez S.R., Rodriguez R.E. Characterization of zebrafish proenkephalin reveals novel opioid sequences. Brain Res. Mol. Brain Res. 114:2003;31-39
    • (2003) Brain Res. Mol. Brain Res. , vol.114 , pp. 31-39
    • Gonzalez, N.V.1    Gonzalez, S.R.2    Rodriguez, R.E.3
  • 10
    • 0030611354 scopus 로고    scopus 로고
    • 7, an endogenous neuropeptide, binds to multiple opioid and nonopioid sites in rat brain
    • 7, an endogenous neuropeptide, binds to multiple opioid and nonopioid sites in rat brain. J. Neurosci. Res. 48:1997;249-258
    • (1997) J. Neurosci. Res. , vol.48 , pp. 249-258
    • Benyhe, S.1    Farkas, J.2    Tóth, G.3    Wollemann, M.4
  • 15
    • 0024516538 scopus 로고
    • Synthesis and biological evaluation of 14-alkoxymorphinans: 2. (-)-N-(cyclopropylmethyl)-4,14-dimethoxymorphinan-6-one, a selective mu opioid receptor antagonist
    • Schmidhammer H., Burkard W.P., Eggstein-Aeppli L., Smith C.F. Synthesis and biological evaluation of 14-alkoxymorphinans: 2. (-)-N-(cyclopropylmethyl)- 4,14-dimethoxymorphinan-6-one, a selective mu opioid receptor antagonist. J. Med. Chem. 32:1989;418-421
    • (1989) J. Med. Chem. , vol.32 , pp. 418-421
    • Schmidhammer, H.1    Burkard, W.P.2    Eggstein-Aeppli, L.3    Smith, C.F.4
  • 16
    • 0023139286 scopus 로고
    • Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonists
    • Portoghese P.S., Lipkowski A.W., Takemori A.E. Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonists. Life Sci. 40:1987;1287-1292
    • (1987) Life Sci. , vol.40 , pp. 1287-1292
    • Portoghese, P.S.1    Lipkowski, A.W.2    Takemori, A.E.3
  • 17
    • 0017036162 scopus 로고
    • Chronic catheterization of the spinal subarachnoid space
    • Yaksh T.L., Rudy T.A. Chronic catheterization of the spinal subarachnoid space. Physiol. Behav. 17:1976;1031-1036
    • (1976) Physiol. Behav. , vol.17 , pp. 1031-1036
    • Yaksh, T.L.1    Rudy, T.A.2
  • 18
    • 0017184389 scopus 로고
    • A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
    • Bradford M.M. A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding. Anal. Biochem. 72:1986;248-254
    • (1986) Anal. Biochem. , vol.72 , pp. 248-254
    • Bradford, M.M.1
  • 21
    • 0032578605 scopus 로고    scopus 로고
    • In vitro binding and signaling profile of the novel μ-opioid receptor agonist endomorphin-2 in rat brain membranes
    • Spetea M., Monory K., Tömböly Cs., Tóth G., Tzavara E., Benyhe S., et al. In vitro binding and signaling profile of the novel μ-opioid receptor agonist endomorphin-2 in rat brain membranes. Biochem. Biophys. Res. Commun. 250:1998;720-725
    • (1998) Biochem. Biophys. Res. Commun. , vol.250 , pp. 720-725
    • Spetea, M.1    Monory, K.2    Tömböly, Cs.3    Tóth, G.4    Tzavara, E.5    Benyhe, S.6
  • 24
    • 0017683782 scopus 로고
    • A synthetic enkephalin analogue with prolonged parenteral and oral analgesic activity
    • Roemer D., Buescher H.H., Hill R.C., Pless J., Bauer W., Cardinaux F., et al. A synthetic enkephalin analogue with prolonged parenteral and oral analgesic activity. Nature. 268:1977;547-549
    • (1977) Nature , vol.268 , pp. 547-549
    • Roemer, D.1    Buescher, H.H.2    Hill, R.C.3    Pless, J.4    Bauer, W.5    Cardinaux, F.6
  • 25
    • 0020527715 scopus 로고
    • Deltakephalin, Tyr-D-Thr-Gly-Phe-Leu-Thr: A new highly potent and fully specific agonist for opiate delta-receptors
    • Zajac J.M., Gacel G., Petit F., Dodey P., Rossignol P., Roques B.P. Deltakephalin, Tyr-D-Thr-Gly-Phe-Leu-Thr: a new highly potent and fully specific agonist for opiate delta-receptors. Biochem. Biophys. Res. Commun. 111:1983;390-397
    • (1983) Biochem. Biophys. Res. Commun. , vol.111 , pp. 390-397
    • Zajac, J.M.1    Gacel, G.2    Petit, F.3    Dodey, P.4    Rossignol, P.5    Roques, B.P.6
  • 27
    • 0033527609 scopus 로고    scopus 로고
    • Antinociceptive effects of endomorphin-1 and -2 in rat
    • Horváth G., Szikszay M., Benedek G. Antinociceptive effects of endomorphin-1 and -2 in rat. Life Sci. 65:1999;2635-2641
    • (1999) Life Sci. , vol.65 , pp. 2635-2641
    • Horváth, G.1    Szikszay, M.2    Benedek, G.3
  • 28
    • 0033916838 scopus 로고    scopus 로고
    • The effects of ketamine and its enantiomers on the morphine- or dexmedetomidine-induced antinociception after intrathecal administration in rats
    • Joó G., Horváth G., Klimscha W., Kékesi G., Dobos I., Szikszay M., et al. The effects of ketamine and its enantiomers on the morphine- or dexmedetomidine-induced antinociception after intrathecal administration in rats. Anesthesiology. 93:2000;231-241
    • (2000) Anesthesiology , vol.93 , pp. 231-241
    • Joó, G.1    Horváth, G.2    Klimscha, W.3    Kékesi, G.4    Dobos, I.5    Szikszay, M.6
  • 29
    • 0034450970 scopus 로고    scopus 로고
    • Endomorphin-1 and endomorphin-2. Pharmacology of the selective endogenous μ-opioid receptor agonists
    • Horváth G. Endomorphin-1 and endomorphin-2. Pharmacology of the selective endogenous μ-opioid receptor agonists. Pharmacol. Ther. 88:2000;437-463
    • (2000) Pharmacol. Ther. , vol.88 , pp. 437-463
    • Horváth, G.1
  • 33
    • 0030007631 scopus 로고    scopus 로고
    • Effect of low pH treatment on opioid peptides binding to their receptors and functional coupling of G-proteins to adenylyl cyclase in the rat spinal cord
    • Reddy P.L., Bhargava H.N. Effect of low pH treatment on opioid peptides binding to their receptors and functional coupling of G-proteins to adenylyl cyclase in the rat spinal cord. Peptides. 17:1996;625-628
    • (1996) Peptides , vol.17 , pp. 625-628
    • Reddy, P.L.1    Bhargava, H.N.2
  • 34
    • 0345599276 scopus 로고    scopus 로고
    • Comparison of [Dmt1]DALDA and DAMGO in binding and G protein activation at μ, δ, and κ opioid receptors
    • Zhao G.M., Qian X., Schiller P.W., Szeto H.H. Comparison of [Dmt1]DALDA and DAMGO in binding and G protein activation at μ, δ, and κ opioid receptors. J. Pharmacol. Exp. Ther. 307:2003;947-954
    • (2003) J. Pharmacol. Exp. Ther. , vol.307 , pp. 947-954
    • Zhao, G.M.1    Qian, X.2    Schiller, P.W.3    Szeto, H.H.4
  • 35
    • 0029417155 scopus 로고
    • Recent advances in molecular recognition and signal transduction of active peptides: Receptors for opioid peptides
    • Kieffer B.L. Recent advances in molecular recognition and signal transduction of active peptides: receptors for opioid peptides. Cell. Mol. Neurobiol. 15:1995;615-635
    • (1995) Cell. Mol. Neurobiol. , vol.15 , pp. 615-635
    • Kieffer, B.L.1
  • 38
    • 0029417219 scopus 로고
    • Adenylylcyclase supersensitization in mu-opioid receptor-transfected Chinese hamster ovary cells following chronic opioid treatment
    • Avidor-Reiss T., Bayewitch M., Levy R., Matus-Leibovitch N., Nevo I., Vogel Z. Adenylylcyclase supersensitization in mu-opioid receptor-transfected Chinese hamster ovary cells following chronic opioid treatment. J. Biol. Chem. 270:1995;29732-29738
    • (1995) J. Biol. Chem. , vol.270 , pp. 29732-29738
    • Avidor-Reiss, T.1    Bayewitch, M.2    Levy, R.3    Matus-Leibovitch, N.4    Nevo, I.5    Vogel, Z.6
  • 39
    • 0030574052 scopus 로고    scopus 로고
    • Expression and pharmacological characterization of the human mu-opioid receptor in the methylotrophic yeast Pichia pastoris
    • Talmont F., Sidobre S., Demange P., Milon A., Emorine L.J. Expression and pharmacological characterization of the human mu-opioid receptor in the methylotrophic yeast Pichia pastoris. FEBS Lett. 394:1996;268-272
    • (1996) FEBS Lett. , vol.394 , pp. 268-272
    • Talmont, F.1    Sidobre, S.2    Demange, P.3    Milon, A.4    Emorine, L.J.5
  • 40
    • 0029856581 scopus 로고    scopus 로고
    • Functional analysis of cloned opioid receptors in transfected cell lines
    • Piros E.T., Hales T.G., Evans C.J. Functional analysis of cloned opioid receptors in transfected cell lines. Neurochem. Res. 21:1996;1277-1285
    • (1996) Neurochem. Res. , vol.21 , pp. 1277-1285
    • Piros, E.T.1    Hales, T.G.2    Evans, C.J.3
  • 41
    • 0030948994 scopus 로고    scopus 로고
    • G proteins and opioid receptor-mediated signalling
    • Standifer K.M., Pasternak G.W. G proteins and opioid receptor-mediated signalling. Cell. Signal. 9:1997;237-248
    • (1997) Cell. Signal. , vol.9 , pp. 237-248
    • Standifer, K.M.1    Pasternak, G.W.2
  • 42
    • 0028986870 scopus 로고
    • 35S]thio)triphosphate binding to membranes from human neuroblastoma SH-SY5Y cells
    • 35S]thio)triphosphate binding to membranes from human neuroblastoma SH-SY5Y cells. Mol. Pharmacol. 47:1995;848-854
    • (1995) Mol. Pharmacol. , vol.47 , pp. 848-854
    • Traynor, J.R.1    Nahorski, S.R.2
  • 43
    • 2142703828 scopus 로고    scopus 로고
    • Synergistic contributions of the functional groups of epinephrine to its affinity and efficacy at the β2 adrenergic receptor
    • Liapakis G., Chan W.C., Papadokostaki M., Javitch J.A. Synergistic contributions of the functional groups of epinephrine to its affinity and efficacy at the β2 adrenergic receptor. Mol. Pharmacol. 65:2004;1181-1190
    • (2004) Mol. Pharmacol. , vol.65 , pp. 1181-1190
    • Liapakis, G.1    Chan, W.C.2    Papadokostaki, M.3    Javitch, J.A.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.