A method for the synthesis of 2-amino-4-fluorobicyclo[3.1.0]hexane-2,6- dicarboxylic acid-[3H2]

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 47, Issue 9, 2004, Pages 571-581

  Kuo, Fengjiun ^a   Kulanthaivel, Palaniappan ^a   Rener, Gregory A ^a   Yi, Ping ^a   Wheeler, William J ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

mGluR agonist; Sodium borotritide reduction; Tritium labeling of secondary alcohol

Indexed keywords

HEXANE; KETONES; TRITIUM;

% REDUCTIONS; DEUTERIUM LABELLING; DICARBOXYLIC ACID; HIGH SPECIFIC ACTIVITIES; LABELINGS; MGLUR AGONIST; PYRIDINIUM TRIBROMIDE; SECONDARY ALCOHOLS; SODIUM BOROTRITIDE REDUCTION; TRITIUM LABELING OF SECONDARY ALCOHOL;

SODIUM;

2 AMINO 4 FLUOROBICYCLO[3.1.0]HEXANE 2,6 DICARBOXYLIC ACID H 3; BOROHYDRIDE SODIUM H 3; BORON DERIVATIVE; CARBOXYLIC ACID DERIVATIVE; GLUTAMATE RECEPTOR AGONIST; KETONE; NICKEL; PYRIDINIUM DERIVATIVE; PYRIDINIUM TRIBORIDE; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

ARTICLE; BROMINATION; DRUG SYNTHESIS; ISOTOPE LABELING; NUCLEAR MAGNETIC RESONANCE; RADIOCHEMISTRY; REACTION ANALYSIS; REDUCTION;

TRITIUM;

EID: 4344701824     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/jlcr.843     Document Type: Article

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