4-Hydroxy-2-quinolones 138. Synthesis and study of structure-biological activity relationships in a series of 1-hydroxy-3-oxo-5,6-dihydro-3H-pyrrolo[3, 2,1-ij]quinoline-2-carboxylic acid anilides

Chemistry of Heterocyclic Compounds

Volumn 43, Issue 12, 2007, Pages 1532-1539

  Ukrainets, I V ^a   Mospanova, E V ^a   Bereznyakova, N L ^a   Naboka, O I ^a  

^a NATIONAL UNIVERSITY OF PHARMACY   (Ukraine)

Author keywords

4 hydroxy 2 oxo 1,2 dihydroquinoline 3 carboxylic acids; Amidation; Anilides; Antitubercular activity; Diuretics

Indexed keywords

EID: 43349087260     PISSN: 00093122     EISSN: 15738353     Source Type: Journal    
DOI: 10.1007/s10593-007-0237-0     Document Type: Article

References (29)

1. I. V. Ukrainets, A. A. Tkach, and M. N. Khomovskaya, Khim. Geterotsikl. Soedin., 1799 (2007).
2. [Chem. Heterocycl. Comp., 43, 1527 (2007)].
3. S. R. Khan, A. Mhaka, R. Pili, and J. T. Isaacs, Bioorg. Med. Chem. Lett., 11, 451 (2001).
4. S. Jönsson, G. Andersson, T. Fex, T. Fristedt, G. Hedlund, K. Jansson, L. Abramo, I. Fritzson, O. Pekarski, A. Runström, H. Sandin, A. Thuvesson, and A. Björk, J. Med. Chem., 47, 2075 (2004).
5. K. Tsuji, G. W. Spears, K. Nakamura, T. Tojo, N. Seki, A. Sugiyama, and M. Matsuo, Bioorg. Med. Chem. Lett., 12, 85 (2002).
6. A. Björk, S. Jönsson, T. Fex, and G. Hedlund, US Patent 6077851 (2000); http://ep.espacenet.com.
7. J. Shi, Z. Xiao, M. A. Ihnat, C. Kamat, B. Pandit, Z. Hu, and P.-K. Li, Bioorg. Med. Chem. Lett., 13, 1187 (2003).
8. J. H. M. Lange, P. C. Verveer, S. J. M. Osnabrug, and G. M. Visser, Tetrahedron Lett., 42, 1367 (2001).
9. I. V. Ukrainets, A. A. Tkach, L. V. Sidorenko, and O. V. Gorokhova, Khim. Geterotsikl. Soedin., 1508 (2006).
10. [Chem. Heterocycl. Comp., 42, 1301 (2006)].
11. I. V. Ukrainets, L. V. Sidorenko, E. N. Svechnikova, and O. V. Shishkin, Khim. Geterotsikl. Soedin., 1503 (2007).
12. [Chem. Heterocycl. Comp., 43, 1275 (2007)].
13. E. Eriksoo, E. N. Sandberg, and L. J. T. Stalhandske, US Patent 4547511 (1985); http://ep.espacenet.com.
14. A. Kutyrev and T. Kappe, J. Heterocycl. Chem., 34, 969 (1997).
15. I. V. Ukrainets, E. V. Mospanova, and L. V. Sidorenko, Khim. Geterotsikl. Soedin., 1023 (2007).
16. [Chem. Heterocycl. Comp., 43, 863 (2007)].
17. I. V. Ukrainets, L. V. Sidorenko, O. V. Gorokhova, S. V. Shiskhina, and A. V. Turov, Khim. Geterotsikl. Soedin., 736 (2007).
18. [Chem. Heterocycl. Comp., 43, 617 (2007)].
19. L. B. Heifets, in: L. B. Heifets (editor), Drug Susceptibility in the Chemotherapy of Mycobacterial Infections, CRC Press, Boca Raton (1991), p. 89.
20. C. B. Inderleid and K. A. Nash, in: V. Lorian (editor), Antibiotics in Laboratory Medicine, Williams and Wilkins, Baltimore (1996), p. 127.
21. Abdel Naser Dakkakh, Dissertations of Candidate in Pharmaceutical Sciences, Kharkiv (2002).
22. I. V. Ukrainets, N. L. Bereznyakova, and E. V. Mospanova, Khim. Geterotsikl. Soedin., 1015 (2007).
23. [Chem. Heterocycl. Comp., 43, 856 (2007)].
24. L. N. Sernov and V. V. Gatsura, Elements of Experimental Pharmacology [in Russian], Moscow (2000), p. 103.
25. N. I. Fadeeva, M. V. Shulgina, and R. G. Glushkov, Khim.-Farm. Zh., 27, No. 5, 4 (1993).
26. I. V. Ukrainets, A. A. Tkach, E. V. Mospanova, and E. N. Svechnikova, Khim. Geterotsikl. Soedin., 1196 (2007)
27. [Chem. Heterocycl. Comp., 43, 1014 (2007)].
28. I. V. Ukrainets, L. V. Sidorenko, O. V. Gorokhova, E. V. Mospanova, and O. V. Shishkin, Khim. Geterotsikl. Soedin., 718 (2006).
29. [Chem. Heterocycl. Comp., 42, 631 (2006)].