Design of high-affinity peptide conjugates with optimized fluorescence quantum yield as markers for small peptide transporter PEPT1 (SLC15A1)

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 8, 2008, Pages 2555-2557

  Bahadduri, Praveen M ^a   Ray, Abhijit ^a   Khandelwal, Akash ^a   Swaan, Peter W ^a  

^a UNIVERSITY OF MARYLAND SCHOOL OF PHARMACY   (United States)

Author keywords

Alexa Fluor 350 ; CoMFA; Fluorescence; High throughput screening; hPEPT1; Peptide conjugation; Transporter

Indexed keywords

GLYCYLSARCOSINE; LYSYLALANINE; LYSYLGLYCINE; LYSYLGLYCYLGLYCINE; LYSYLSERINE; LYSYLVALINE; MONOCARBOXYLATE TRANSPORTER 1; PEPTIDE TRANSPORTER 1; TRITIUM; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CHO CELL; COMPARATIVE MOLECULAR FIELD ANALYSIS; CONTROLLED STUDY; FLUORESCENCE; HIGH THROUGHPUT SCREENING; NONHUMAN; QUANTITATIVE STRUCTURE ACTIVITY RELATION; QUANTUM YIELD;

ANIMALS; CHO CELLS; CRICETINAE; CRICETULUS; DRUG DESIGN; FLUORESCENT DYES; HUMANS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PEPTIDES; SYMPORTERS;

ALEXA;

EID: 41849116361     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.03.044     Document Type: Article

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