Pharmacokinetics of diclofenac and its interaction with enrofloxacin in sheep

Research in Veterinary Science

Volumn 84, Issue 3, 2008, Pages 452-456

  Rahal, Anu ^c   Kumar, Amit ^b   Ahmad, A H ^c   Malik, J K ^a  

^a INDIAN VETERINARY RESEARCH INSTITUTE   (India)

^b U P State Govt ^*  (India)

^c G B PANT UNIVERSITY OF AGRICULTURE AND TECHNOLOGY   (India)

Author keywords

Diclofenac; Enrofloxacin; Intramuscular; Pharmacokinetics; Sheep

Indexed keywords

3 D VET; CYTOCHROME P450; DICLOFENAC; ENROFLOXACIN; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; AREA UNDER THE CURVE; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DISTRIBUTION VOLUME; DOSE CALCULATION; DRUG ABSORPTION; DRUG BIOAVAILABILITY; DRUG BLOOD LEVEL; DRUG CLEARANCE; DRUG DETERMINATION; DRUG DOSE REGIMEN; DRUG ELIMINATION; DRUG HALF LIFE; ENZYME INHIBITION; FEMALE; LOADING DRUG DOSE; MAXIMUM PLASMA CONCENTRATION; MEAN RESIDENCE TIME; NONHUMAN; PLASMA CONCENTRATION-TIME CURVE; RECOMMENDED DRUG DOSE; SHEEP; SINGLE DRUG DOSE; TIME TO MAXIMUM PLASMA CONCENTRATION;

ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; DICLOFENAC; DRUG INTERACTIONS; FLUOROQUINOLONES; INJECTIONS, INTRAMUSCULAR; INJECTIONS, INTRAVENOUS; KINETICS; SHEEP;

OVIS ARIES;

EID: 41749104853     PISSN: 00345288     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.rvsc.2007.06.002     Document Type: Article

References (26)

1. Ahangar A.H., and Srivastava A.K. Pharmacokinetics of enrofloxacin in febrile crossbred bovine calves. Indian Journal of Pharmacology 32 (2000) 305-308
2. Altreuher, P., 1987. Safety and tolerance of enrofloxacin in dogs and cats. In: Proc. First Int. Baytril Symp., Bonn., Germany. Cited from Enrofloxacin Revisited" 1994. Vet. Med. 744-753.
3. Averginos A., Karidas T., and Malamataris S. Extractionless high performance liquid chromatographic method for the determination of diclofenac in human plasma and urine. Journal of Chromatography 619 (1993) 324-329
4. Calabro J.J. Eficacy of diclofenac in anklyosing spondylitis. American Journal of Medicine 80 (1986) 58-64
5. Dudley M.N. Pharmacodynamics and pharmacokinetics of antibiotics with special reference to the fluoroquinolones. Am. J. Med. 91 suppl 6A (1991) 455-505
6. Gibaldi M., and Perrier D. Pharmacokinetics (1982), Marcel Dekker, New York
7. Jairam, R., Gatne, M.M., Somkuwar, A.P., Jagadish, S., Ranade, V.V., 1995. Pharmacokinetics of Nonsteroidal anti-inflammatory drug, Clogil (diclofenac sodium) in buffalo calves. Abstract in IInd National Convention of Veterinary Pharmacology and Toxicology.
8. John V.A. The pharmacokinetics of diclofenac (Voltarol) in animals and man. Rheumatology and Rehabilitation 2 (1979) 22-35
9. Joly V., Pangon B., Brion N., Vallois J.M., and Carbon C. Enhancement of the therapeutic effect of cephalosporins in experimental endocarditis by altering their pharmacokinetics with diclofenac. Journal of Veterinary Pharmacology and Therapeutics 246 (1988) 695-700
10. Kumar N., Singh S.D., and Jayachandran C. Pharmacokinetic studies of diclofenac and its interaction with enrofloxacin in buffalo calves. Journal of Veterinary Sciences 4 (2003) 155-159
11. Martinez M.N. Use of pharmacokinetics in veterinary medicine. Article I: Noncompartmental methods of drug characterization: statistical moment theory. Journal of American Veterinary and Medical Association 213 (1998) 974-980
12. Martinez M.N. Use of pharmacokinetics in veterinary medicine. Article II: Volume, clearance and half-life. Journal of American Veterinary and Medical Association 213 (1998) 1122-1127
13. Menasse R., Hedwall P.R., Kraetz J., Pesicin C., Riesterer L., Sallamann Z.R., and Jaques R. Pharmacological properties of diclofenac and its metabolites. Scandinavian Journal of Rheumatology 22 (1978) 5-16
14. Mueller E.A., Kovarike J.M., Koelle E.U., Merdjan H., Johnston A., and Hitzenbeger G. Pharmacokinetics of cyclosporine and multiple-dose diclofenac during coadministration. Journal of Clinical Pharmacology 33 (1993) 936-943
15. Nakashi S., and Okuno H. Comparison of inhibitory effects of new quinolones on drug metabolizing activity in the liver. Japanese Journal of Pharmacology 53 (1990) 81-96
16. Nergelius G., Vinge E., Bentsson H.I., Bjorkman R., and Gurbb A. No effect of diclofenac on the pharmacokinetics of cloxacillin. Pharmacology and Toxicology 81 (1997) 26-30
17. Nielsen P., and Gyrd-Hansen N. Bioavailability of enrofloxacin after oral administration to fed and fasted pigs. Pharmacology and Toxicology 80 (1997) 246-250
18. Sano M., Kawakatsu K., Ohkita C., et al. Effects of enoxacin, ofloxacin and norfloxacin on theophylline disposition in humans. European Journal of Clinical Pharmacology 35 (1988) 161-165
19. Shlosberg A., Ershov E., Bellaiche M., Hanji V., Weisman Y., and Soback S. The inhibitory effects of the fluoroquinolone antimicrobials norfloxacin and enrofloxacin on hepatic microsomal cytochrome P-450 monooxygenases in broiler chickens. Drug Metabolism Drug Interaction 14 2 (1997) 109-122
20. Struck H.G., Bariszlovich A., Kuhlmann O., and WEISS M. Concentration of diclofenac in aqueous humor and in plasma after IV injections in 59 patients undergoing cataract surgery. Klin. Monatsbl Augenheilkd 218 (2001) 85-88
21. Tang W., Stearns R.A., Kwei G.Y., Iliff S.A., Miller R.R., Egan M.A., Yu N.X., Dean D.C., Kumar S., Shou M., Lin J.H., and Baille T.A. Interaction of diclofenac and quinidine in monkey: stimulation of diclofenac metabolism. Journal of Pharmacology and Experimental Therapeutics 291 (1999) 1068-1074
22. Torres-Lopez J.E., Lopez-Munoz F.J., Costanera-Hernandez G., Flores-Murrieta F.J., and Granados-Soto V. Pharmacokinetic-Pharmacodynamic modelling of the antinociceptive effect of diclofenac in the rat. Journal of Pharmacology and Experimental Therapeutics 291 (1997) 1068-1074
23. Tsuchiya T., Terakawa K., Ishibashi K., Shibuya T., and Fugimura H. Disposition and enterohepatic circulation of diclofenac in dogs. Drug Research 30 (1980) 1650-1653
24. Varma, R., Ahmad, A.H., Sharma, L.D., 2000. Pharmacokinetics of enrofloxacin and its interaction with diclofenac sodium in cattle. Compendium of abstracts. In: First National Annual Conference of Indian Society of Veterinary Pharmacology and Toxicology, pp. 48.
25. Wagner J., and Sulc M. Binding of diclofenac-sodium(Voltaren) to serum proteins of different species and interactions with other drugs in protein binding. Aktuelle Rheumatologie 4 (1979) 153
26. Willis J.V., Kendall M.J., Flinn R.M., Thornill D., and Welling P.G. The pharmacokinetics of diclofenac sodium after intravenous or oral administration. European Journal of Clinical Pharmacology 16 (1979) 405-410