Pharmacophore identification of Raf-1 kinase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 7, 2008, Pages 2346-2350

  Zhu, Tian ^a   Jiao, Yu ^a   Chen, Ya Dong ^a   Wang, Xuan ^a   Li, Hui Fang ^a   Zhang, Lu Yong ^a   Lu, Tao ^a  

^a CHINA PHARMACEUTICAL UNIVERSITY   (China)

Author keywords

Docking; Homology modeling; Pharmacophore; Raf 1 kinase

Indexed keywords

HYDROGEN; PHOSPHOTRANSFERASE INHIBITOR; RAF PROTEIN;

ARTICLE; CORRELATION COEFFICIENT; DRUG DESIGN; DRUG SCREENING; HYDROGEN BOND; HYDROPHOBICITY; MODEL; PHARMACOPHORE;

BINDING SITES; BIOLOGICAL TRANSPORT; ENZYME INHIBITORS; HYDROGEN BONDING; HYDROPHOBICITY; MODELS, BIOLOGICAL; MODELS, CHEMICAL; PROTO-ONCOGENE PROTEINS C-RAF; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 41149091871     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.02.068     Document Type: Article

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