Synthesis and biological evaluation of novel 8-aminomethylated oroxylin A analogues as α-glucosidase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 5, 2008, Pages 1659-1662

  Hari Babu, T ^a   Rama Subba Rao, V ^a   Tiwari, Ashok K ^a   Suresh Babu, K ^a   Srinivas, P V ^a   Ali, Amtul Z ^a   Madhusudana Rao, J ^a  

^a INDIAN INSTITUTE OF CHEMICAL TECHNOLOGY   (India)

Author keywords

Mannich reaction; Oroxylin A; Oroxylum indicum; Primary amines; Secondary amines; Glucosidase inhibition

Indexed keywords

4 FORMALDEHYDE; 8 AMINOMETHYLATED OROXYLIN A DERIVATIVE; ALPHA GLUCOSIDASE INHIBITOR; AMINE; BAICALEIN; CHRYSIN; FORMALDEHYDE; OROXYLIN A; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; ENZYME INHIBITION; IC 50; MANNICH REACTION; NONHUMAN; RAT; SYNTHESIS; YEAST;

OROXYLUM INDICUM; RATTUS;

EID: 39849111649     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.01.055     Document Type: Article

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