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Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 5, 2008, Pages 1681-1687

Thiol-based angiotensin-converting enzyme 2 inhibitors: P1′ modifications for the exploration of the S1′ subsite

(4) Deaton, David N a Graham, Kevin P a Gross, Jeffrey W a Miller, Aaron B a

a GLAXOSMITHKLINE (United States)

Author keywords

Angiotensin converting enzyme 2; Metalloproteases; Protease inhibitors; Thiols

Indexed keywords

ANGIOTENSIN CONVERTING ENZYME 2; CARBENE; DIPEPTIDYL CARBOXYPEPTIDASE INHIBITOR; MALACHITE GREEN; METALLOPROTEINASE INHIBITOR; MLN 4760; PHENYL GROUP; PHENYLALANINE DERIVATIVE; THIOL GROUP; TYROSINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL MEMBRANE PERMEABILITY; CHEMICAL MODIFICATION; DRUG METABOLISM; DRUG POTENCY; DRUG POTENTIATION; ENZYME INHIBITION; HYDROGEN BOND; IN VITRO STUDY; NONHUMAN; STRUCTURE ACTIVITY RELATION;

EID: 39849104176 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2008.01.046 Document Type: Article

Times cited : (3)

References (21)

1
- 0038053724
- M. Donoghue F. Hsieh E. Baronas K. Godbout M. Gosselin N. Stagliano M. Donovan B. Woolf K. Robison R. Jeyaseelan R.E. Breitbart S. Acton Circ. Res. 87 2000 e1
- (2000) Circ. Res. , vol.87 , pp. e1
- Donoghue, M.¹ Hsieh, F.² Baronas, E.³ Godbout, K.⁴ Gosselin, M.⁵ Stagliano, N.⁶ Donovan, M.⁷ Woolf, B.⁸ Robison, K.⁹ Jeyaseelan, R.¹⁰ Breitbart, R.E.¹¹ Acton, S.¹²

2
- 0034721906
- S.R. Tipnis N.M. Hooper R. Hyde E. Karran G. Christie A.J. Turner J. Biol. Chem. 275 2000 33238
- (2000) J. Biol. Chem. , vol.275 , pp. 33238
- Tipnis, S.R.¹ Hooper, N.M.² Hyde, R.³ Karran, E.⁴ Christie, G.⁵ Turner, A.J.⁶

3
- 33645299090
- U. Danilczyk J.M. Penninger Circ. Res. 98 2006 463
- (2006) Circ. Res. , vol.98 , pp. 463
- Danilczyk, U.¹ Penninger, J.M.²

4
- 33646352935
- K. Kuba Y. Imai J.M. Penninger Curr. Opin. Pharm. 6 2006 271
- (2006) Curr. Opin. Pharm. , vol.6 , pp. 271
- Kuba, K.¹ Imai, Y.² Penninger, J.M.³

5
- 33646538118
- E.A. Tallant C.M. Ferrario P.E. Gallagher Future Cardiol. 2 2006 335
- (2006) Future Cardiol. , vol.2 , pp. 335
- Tallant, E.A.¹ Ferrario, C.M.² Gallagher, P.E.³

6
- 0037142101
- M.A. Crackower R. Sarao G.Y. Oudit C. Yagil I. Kozieradzki S.E. Scanga A.J. Oliveira-dos-Santos J. da Costa L. Zhang Y. Pei J. Scholey C.M. Ferrario A.S. Manoukian M.C. Chappell P.H. Backx Y. Yagil J.M. Penninger Nature 417 2002 822
- (2002) Nature , vol.417 , pp. 822
- Crackower, M.A.¹ Sarao, R.² Oudit, G.Y.³ Yagil, C.⁴ Kozieradzki, I.⁵ Scanga, S.E.⁶ Oliveira-dos-Santos, A.J.⁷ da Costa, J.⁸ Zhang, L.⁹ Pei, Y.¹⁰ Scholey, J.¹¹ Ferrario, C.M.¹² Manoukian, A.S.¹³ Chappell, M.C.¹⁴ Backx, P.H.¹⁵ Yagil, Y.¹⁶ Penninger, J.M.¹⁷

7
- 33746724157
- S.B. Gurley A. Allred T.H. Le R. Griffiths L. Mao N. Philip T.A. Haystead M. Donoghue R.E. Breitbart S.L. Acton H.A. Rockman T.M. Coffman J. Clin. Invest. 116 2006 2218
- (2006) J. Clin. Invest. , vol.116 , pp. 2218
- Gurley, S.B.¹ Allred, A.² Le, T.H.³ Griffiths, R.⁴ Mao, L.⁵ Philip, N.⁶ Haystead, T.A.⁷ Donoghue, M.⁸ Breitbart, R.E.⁹ Acton, S.L.¹⁰ Rockman, H.A.¹¹ Coffman, T.M.¹²

8
- 33645834948
- K. Yamamoto M. Ohishi T. Katsuya N. Ito M. Ikushima M. Kaibe Y. Tatara A. Shiota S. Sugano S. Takeda H. Rakugi T. Ogihara Hypertension 47 2006 718
- (2006) Hypertension , vol.47 , pp. 718
- Yamamoto, K.¹ Ohishi, M.² Katsuya, T.³ Ito, N.⁴ Ikushima, M.⁵ Kaibe, M.⁶ Tatara, Y.⁷ Shiota, A.⁸ Sugano, S.⁹ Takeda, S.¹⁰ Rakugi, H.¹¹ Ogihara, T.¹²

9
- 33744731510
- G.Y. Oudit A.M. Herzenberg Z. Kassiri D. Wong H. Reich R. Khokha M.A. Crackower P.H. Backx J.M. Penninger J.W. Scholey Am. J. Pathol. 168 2006 1808
- (2006) Am. J. Pathol. , vol.168 , pp. 1808
- Oudit, G.Y.¹ Herzenberg, A.M.² Kassiri, Z.³ Wong, D.⁴ Reich, H.⁵ Khokha, R.⁶ Crackower, M.A.⁷ Backx, P.H.⁸ Penninger, J.M.⁹ Scholey, J.W.¹⁰

10
- 85120133738
- Acton, S. L.; Ocain, T. D.; Gould, A. E.; Dales, N. A.; Guan, B.; Brown, J. A.; Patane, M.; Kadambi, V. J.; Solomon, M.; Stricker-Krongrad, A. PCT Int. Appl. WO 039997, 2002 ; Chem. Abstr . 2002 , 136 , 402027.

11
- 0344395657
- W. Li M.J. Moore N. Vasilieva J. Sui S.K. Wong M.A. Berne M. Somasundaran J.L. Sullivan K. Luzuriaga T.C. Greenough H. Choe M. Farzan Nature 426 2003 450
- (2003) Nature , vol.426 , pp. 450
- Li, W.¹ Moore, M.J.² Vasilieva, N.³ Sui, J.⁴ Wong, S.K.⁵ Berne, M.A.⁶ Somasundaran, M.⁷ Sullivan, J.L.⁸ Luzuriaga, K.⁹ Greenough, T.C.¹⁰ Choe, H.¹¹ Farzan, M.¹²

12
- 23844463115
- K. Kuba Y. Imai S. Rao H. Gao F. Guo B. Guan Y. Huan P. Yang Y. Zhang W. Deng L. Bao B. Zhang G. Liu Z. Wang M. Chappell Y. Liu D. Zheng A. Leibbrandt T. Wada A.S. Slutsky D. Liu C. Qin C. Jiang J.M. Penninger Nat. Med. 11 2005 875
- (2005) Nat. Med. , vol.11 , pp. 875
- Kuba, K.¹ Imai, Y.² Rao, S.³ Gao, H.⁴ Guo, F.⁵ Guan, B.⁶ Huan, Y.⁷ Yang, P.⁸ Zhang, Y.⁹ Deng, W.¹⁰ Bao, L.¹¹ Zhang, B.¹² Liu, G.¹³ Wang, Z.¹⁴ Chappell, M.¹⁵ Liu, Y.¹⁶ Zheng, D.¹⁷ Leibbrandt, A.¹⁸ Wada, T.¹⁹ Slutsky, A.S.²⁰ more..

13
- 34248597758
- I. Hamming M.E. Cooper B.L. Haagmans N.M. Hooper R. Korstanje A.D.M.E. Osterhaus W. Timens A.J. Tumer G. Navis H. van Goor J. Pathol. 212 2007 1
- (2007) J. Pathol. , vol.212 , pp. 1
- Hamming, I.¹ Cooper, M.E.² Haagmans, B.L.³ Hooper, N.M.⁴ Korstanje, R.⁵ Osterhaus, A.D.M.E.⁶ Timens, W.⁷ Tumer, A.J.⁸ Navis, G.⁹ van Goor, H.¹⁰

14
- 0037048716
- N.A. Dales A.E. Gould J.A. Brown E.F. Calderwood B. Guan C.A. Minor J.M. Gavin P. Hales V.K. Kaushik M. Stewart P.J. Tummino C.S. Vickers T.D. Ocain M.A. Patane J. Am. Chem. Soc. 124 2002 11852
- (2002) J. Am. Chem. Soc. , vol.124 , pp. 11852
- Dales, N.A.¹ Gould, A.E.² Brown, J.A.³ Calderwood, E.F.⁴ Guan, B.⁵ Minor, C.A.⁶ Gavin, J.M.⁷ Hales, P.⁸ Kaushik, V.K.⁹ Stewart, M.¹⁰ Tummino, P.J.¹¹ Vickers, C.S.¹² Ocain, T.D.¹³ Patane, M.A.¹⁴

15
- 0037507256
- L. Huang D.J. Sexton K. Skogerson M. Devlin R. Smith I. Sanyal T. Parry R. Kent J. Enright Q. Wu G. Conley D. DeOliveira L. Morganelli M. Ducar C.R. Wescott R.C. Ladner J. Biol. Chem. 278 2003 15532
- (2003) J. Biol. Chem. , vol.278 , pp. 15532
- Huang, L.¹ Sexton, D.J.² Skogerson, K.³ Devlin, M.⁴ Smith, R.⁵ Sanyal, I.⁶ Parry, T.⁷ Kent, R.⁸ Enright, J.⁹ Wu, Q.¹⁰ Conley, G.¹¹ DeOliveira, D.¹² Morganelli, L.¹³ Ducar, M.¹⁴ Wescott, C.R.¹⁵ Ladner, R.C.¹⁶

16
- 33646256792
- M. Rella C.A. Rushworth J.L. Guy A.J. Turner T. Langer R.M. Jackson J. Chem. Inf. Model 46 2006 708
- (2006) J. Chem. Inf. Model , vol.46 , pp. 708
- Rella, M.¹ Rushworth, C.A.² Guy, J.L.³ Turner, A.J.⁴ Langer, T.⁵ Jackson, R.M.⁶

17
- 9644258512
- M.J. Huentelman J. Zubcevic J.A. Hernandez Prada X. Xiao D.S. Dimitrov M.K. Raizada D.A. Ostrov Hypertension 44 2004 903
- (2004) Hypertension , vol.44 , pp. 903
- Huentelman, M.J.¹ Zubcevic, J.² Hernandez Prada, J.A.³ Xiao, X.⁴ Dimitrov, D.S.⁵ Raizada, M.K.⁶ Ostrov, D.A.⁷

18
- 38149094270
- D.N. Deaton E.N. Gao K.P. Graham J.W. Gross A.B. Miller J.M. Strelow Bioorg. Med. Chem. Lett. 18 2008 732
- (2008) Bioorg. Med. Chem. Lett. , vol.18 , pp. 732
- Deaton, D.N.¹ Gao, E.N.² Graham, K.P.³ Gross, J.W.⁴ Miller, A.B.⁵ Strelow, J.M.⁶

19
- 0032949615
- J.D. Irvine L. Takahashi K. Lockhart J. Cheong J.W. Tolan H.E. Selick J.R. Grove J. Pharm. Sci. 88 1999 28
- (1999) J. Pharm. Sci. , vol.88 , pp. 28
- Irvine, J.D.¹ Takahashi, L.² Lockhart, K.³ Cheong, J.⁴ Tolan, J.W.⁵ Selick, H.E.⁶ Grove, J.R.⁷

20
- 85120109043
- M.H. Lambert P.S. Charifson Practical Application of Computer-Aided Drug Design 1997 Marcel Dekker New York, NY 243
- (1997) , pp. 243
- Lambert, M.H.¹

21
- 2342418543
- P. Towler B. Staker S.G. Prasad S. Menon J. Tang T. Parsons D. Ryan M. Fisher D. Williams N.A. Dales M.A. Patane M.W. Pantoliano J. Biol. Chem. 279 2004 17996
- (2004) J. Biol. Chem. , vol.279 , pp. 17996
- Towler, P.¹ Staker, B.² Prasad, S.G.³ Menon, S.⁴ Tang, J.⁵ Parsons, T.⁶ Ryan, D.⁷ Fisher, M.⁸ Williams, D.⁹ Dales, N.A.¹⁰ Patane, M.A.¹¹ Pantoliano, M.W.¹²

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