Cycloaddition reactions with 2,3-benzodiazepine derivatives

Journal of Heterocyclic Chemistry

Volumn 44, Issue 2, 2007, Pages 431-435

  Kertész, Máriusz ^a   Pallagi, István ^a   Sólyom, Sándor ^a  

^a TEVA PHARMACEUTICALS   (Israel)

Author keywords

[No Author keywords available]

Indexed keywords

BENZODIAZEPINE DERIVATIVE; CARBON; DIAZOMETHANE; NITRILE OXIDE; NITROGEN;

ADDITION REACTION; ARTICLE; CHEMICAL REACTION; CYCLOADDITION; EXPERIMENTAL STUDY; NONHUMAN;

EID: 36749095135     PISSN: 0022152X     EISSN: None     Source Type: Journal    
DOI: 10.1002/jhet.5570440224     Document Type: Article

References (12)

1. Parsons, G. C.; Danysz, W.; Quack, G. Drug News Perspect, 1988, 11, 523.
2. De Sarro, G.; Gitto, R.; Russo, E. Ibbadu, G. F.; Bareca, M. L.; Chimirri, A. Curr. Top. Med. Chem. 2005, 5, 31.
3. Sólyom, S.; Tarnawa, I. Curr. Pharm. Design 2002, 8, 913.
4. Sólyom, S.; Ábrah́am, G.; Hámori, T.; Berzsenyi, P.; Andrási, F.; Kurucz, I. PCT Int. Appl. WO 2004069197, Chem. Abstr. 2004, 141, 174197.
5. Mukaiyama, T.; Hoshino, T. J. Am. Chem. Soc., 1960, 82, 5339.
6. Andrási, F.; Berzsenyi, P.; Botka, P.; Farkas, S.; Goldschmidt, K.; Hámori, T.; Korösi, J.; Moravcsik I.; Tarnawa, I. Eur. Pat. Appl. EP 492,485, Chem. Abstr. 1992, 117, 171478.
7. De Sarro, G.; Chimirri, A.; De Sarro, A.; Gitto, R.; Grasso, S.; Giusti, P.; Chapman, A. G. Eur. J. Pharm., 1995, 294, 411.
8. Vyas, D. M.; Chiang, Y.; Doyle, T. W. Tetrahedron Lett. 1984, 25, 487.
9. Csuzdi, E.; Migléczi, K.; Hazai, I.; Berzsenyi, P.; Pallagi, I.; Horváth, Gy.; Lengyel, Gy., Sólyom, S. Bioorg. Med. Chem. Lett. 2005, 15, 4662.
10. 50 μM.)
11. Swinyard, B. A. J. Pharmacol. Exp. Ther. 1952, 106, 319. (10 mice/dose and 3-4 doses were used; 60 min pretreatment po).
12. Randall, L. O.; Schalleck, W.; Heise, G. A.; Keth, E. F.; Bagdon, R. E. J. Pharmacol. Exp. Ther. 1960, 129, 163. (10 mice/dose and 3-4 doses were used, 30 min pretreatment ip).