A novel short and efficient synthetic route to the antimalarial agent FR900098 and derivatives

Synthesis

Volumn , Issue 22, 2007, Pages 3553-3557

  Perruchon, Johann ^a   Ortmann, Regina ^a   Schlitzer, Martin ^a  

^a PHILIPPS UNIVERSITY MARBURG   (Germany)

Author keywords

Drugs; Multicomponent reactions; Phosphonic acid; Sulfonamides; Sulfones

Indexed keywords

ANTIMALARIAL AGENT FR900098; ONE-POT SYNTHESIS; PHOSPHONIC ACID; SULFONAMIDES; SULFONES;

AMIDES; CARBOXYLIC ACIDS; DERIVATIVES; DRUG THERAPY;

MALARIA CONTROL;

3 (N ACETYL N HYDROXYAMINO)PROPYLPHOSPHONIC ACID; 3 [CETYL(BENZYLOXY)AMINO]PROPANE 1 SULFONYL CHLORIDE; ACETAMIDE DERIVATIVE; ANTIMALARIAL AGENT; DIBENZYL [3 [ACETYL(BENZYLOXY)AMINO]PROPYL]PHOSPHONATE; DIBENZYL PHOSPHONATE; N (BENZYLOXY) N (IODOPROPYL)ACETAMIDE; N (BENZYLOXY) N [3 (METHYLSULFAMOYL)PROPYL]ACETAMIDE; N (BENZYLOXY) N [3 (METHYLSULFANYL)PROPYL]ACETAMIDE; N (BENZYLOXY) N [METHYLSULFONYL)PROPYL]ACETAMIDE; N HYDROXY N [3 (METHYLSULFAMOYL)PROPYL]ACETAMIDE; N HYDROXY N [3 (METHYLSULFONYL)PROPYL]ACETAMIDE; SODIUM 3 [ACETYL(BENZYLOXY)AMINO]PROPANE 1 SULFONATE; SODIUM 3 [ACETYL(HYDROXY)AMINO]PROPANE 1 SULFONATE; SULFONAMIDE; SULFONIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY;

EID: 36749083988     PISSN: 00397881     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-2007-990811     Document Type: Article

References (6)

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