Novel non-PEG derived polyethers as solid supports. 2. Solid-phase synthesis studies

Journal of Combinatorial Chemistry

Volumn 9, Issue 6, 2007, Pages 1012-1027

  Cavalli, Gabriel ^a,c   Shooter, Andrew G ^b   Pears, David A ^b,d   Wellings, Donald A ^b,e   Gulzar, Saeed ^b,e   Steinke, Joachim H G ^a  

^a IMPERIAL COLLEGE LONDON   (United Kingdom)

^b Avecia Biologics Limited   (United Kingdom)

^c UNIVERSITY OF SURREY   (United Kingdom)

^d Reaxa Ltd   (United Kingdom)

^e Chromatide Ltd   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

AGENTS INTERACTING WITH TRANSMITTER, HORMONE OR DRUG RECEPTORS; ALKENE; ETHER DERIVATIVE; LEUCINE ENKEPHALIN; MACROGOL DERIVATIVE; OSMIUM TETRAOXIDE; OXIME; POLY(METHYL METHACRYLATE); RESIN; SOLVENT;

ARTICLE; CHEMICAL MODEL; CHEMISTRY; HYDROXYLATION; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; SYNTHESIS;

ALKENES; ENKEPHALIN, LEUCINE; ETHERS; HYDROXYLATION; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, CHEMICAL; NEUROTRANSMITTER AGENTS; OSMIUM TETROXIDE; OXIMES; POLYETHYLENE GLYCOLS; POLYMETHYL METHACRYLATE; RESINS, SYNTHETIC; SOLVENTS;

EID: 36649008710     PISSN: 15204766     EISSN: None     Source Type: Journal    
DOI: 10.1021/cc7000887     Document Type: Article

References (41)

1. Cavalli, G.; Shooter, A. G.; Pears, D. A.; Steinke, J. H. G. J. Comb. Chem. 2003, 5, 637-644.
2. Porres, L.; Deleuze, H.; Landais, Y. J. Chem. Soc., Perkin Trans. 1 2002, 2198-2203.
3. Fields, G. B.; Fields, C. G. J. Am. Chem. Soc. 1991, 113, 4202-4207.
4. Han, H.; Janda, K. D. Angew. Chem., Int. Ed. 1997, 36, 1731-1733.
5. Meldal, M. Methods Enzymol 1997, 289, 83-104.
6. Czarnik, A. W. Biotechnol. Bioeng. 1998, 61, 77-79.
7. Riedl, R.; Tappe, R.; Berkessel, A. J. Am. Chem. Soc. 1998, 120, 8994-9000.
8. Santini, R.; Griffith, M. C.; Qi, M. Tetrahedron Lett. 1998, 39, 8951-8954.
9. Hudson, D. J. Comb. Chem. 1999, 1, 333-360.
10. Hudson, D. J. Comb. Chem. 1999, 1, 403-457.
11. Vaino, A. R.; Goodin, D. B.; Janda, K. D. J. Comb. Chem. 2000, 2, 330-336.
12. Vaino, A. R.; Janda, K. D. J. Comb. Chem. 2000, 2, 579-596.
13. Hodge, P. Chem. Soc. Rev. 1997, 26, 417-424.
14. Kolb, H. C.; VanNieuwenhze, M. S.; Sharpless, K. B. Chem. Rev. 1994, 94, 2483-2547.
15. Rice, K. D.; Nuss, J. M. Bioorg. Med. Chem. Lett. 2001, 11, 753-755.
16. Cheng, J.-F.; Mjalli, A. M. M. Tetrahedron Lett. 1998, 39, 939-942.
17. Haap, W. J.; Kaiser, D.; Walk, T. B.; Jung, G. Tetrahedron 1998, 54, 3705-3724.
18. Hinzen, B.; Ley, S. V. J. Chem. Soc.-Perkin Trans. 1 1998, 1-2.
19. Shankar, B. B.; Yang, D. Y.; Girton, S.; Ganguly, A. K. Tetrahedron Lett. 1998, 39, 2447-2448.
20. Atherton, E.; Clive, D. L. J.; Sheppard, R. C. J. Am. Chem. Soc. 1975, 97, 6584-6585.
21. Arshady, R.; Atherton, E.; Clive, D. L. J.; Sheppard, R. C. J. Chem. Soc., Perkin Trans. 1 1981, 529-537.
22. Atherton, E.; Logan, C. J.; Sheppard, R. C. J. Chem. Soc., Perkin Trans. 1 1981, 538-546.
23. Wellings, D. A.; Atherton, E. Methods Enzymol. 1997, 289, 44-67.
24. Osby, J. O.; Martin, M. G.; Ganem, B. Tetrahedron Lett. 1984, 25, 2093.
25. Small, P. W.; Sherrington, D. C. J. Chem. Soc., Chem. Commun. 1989, 1589-1591.
26. Colombo, R.; Atherton, E.; Sheppard, R. C.; Woolley, V. Int. J. Pept. Protein Res. 1983, 21, 118-126.
27. Coffey, A. F.; Johnson, T. Int. J. Pept. Protein Res. 1992, 59, 419-430.
28. Englebretsen, D. R.; Harding, D. R. K. Int. J. Pept. Protein Res. 1992, 40, 487-96.
29. Epton, R.; Goddard, P.; Ivin, K. J. Polymer 1980, 21, 1367-1371.
30. Songster, M. F.; Barany, G. Methods Enzymol. 1997, 289, 126-174.
31. Epton, R.; Williams, A. Int. J. Biol. Macromol. 1981, 3, 334-336.
32. Zalipsky, S.; Albericio, P.; Barany, G. Pept.: Struct. Funct., Proc. Am. Pept. Symp., 9th 1985, 257-260.
33. Wells, N. J.; Basso, A.; Bradley, M. Biopolymers 1998, 47, 381-396.
34. Merrifield, R. B. J. Am. Chem. Soc. 1963, 85, 2149-54.
35. Yan, B. Comb. Chem. High Throughput Screen. 1998, 1, 215-229.
36. Hori, M.; Gravert, D. J.; Wentworth, P., Jr.; Janda, K. D. Bioorg. Med. Chem. Lett. 1998, 8, 2363-2368.
37. Alonso, C.; Nantz, M. H.; Kurth, M. J. Tetrahedron Lett. 2000, 41, 5617-5622.
38. Kobayashi, S.; Akiyama, R. Tetrahedron Lett. 1998, 39, 9211-9214.
39. Henderson A. J. PhD Thesis, University of Cambridge, Cambridge, 1999.
40. Avecia Ltd., in-house recipe.
41. Avecia Ltd., in-house recipe.