Preparation of an extended-release matrix tablet using chitosan/Carbopol interpolymer complex

International Journal of Pharmaceutics

Volumn 347, Issue 1-2, 2008, Pages 39-44

  Park, Sung Hyun ^a   Chun, Myung Kwan ^a   Choi, Hoo Kyun ^a  

^a Chosun University   (South Korea)

Author keywords

Carbopol; Chitosan; Extended release; Interpolymer complex

Indexed keywords

AMINE; CARBOXYLIC ACID; CHITOSAN CARBOPOL INTERPOLYMER COMPLEX; COPOLYMER; UNCLASSIFIED DRUG;

ACIDITY; ARTICLE; CONTROLLED DRUG RELEASE; DIFFERENTIAL SCANNING CALORIMETRY; DRUG SYNTHESIS; ELECTRICITY; INFRARED SPECTROSCOPY; PRIORITY JOURNAL; PROTON TRANSPORT; TABLET FORMULATION; THERMAL ANALYSIS; TURBIDIMETRY;

ACRYLATES; BIOLOGICAL AVAILABILITY; CALORIMETRY, DIFFERENTIAL SCANNING; CHITOSAN; DELAYED-ACTION PREPARATIONS; EXCIPIENTS; HYDROGEN-ION CONCENTRATION; KINETICS; METHYLCELLULOSE; MOLECULAR WEIGHT; NEPHELOMETRY AND TURBIDIMETRY; POLYMERS; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; TABLETS; THEOPHYLLINE; WATER;

EID: 36549061102     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2007.06.024     Document Type: Article

References (25)

1. Betageri G.V., Deshmukh D.V., and Gupta R.B. Oral sustained release bioadhesive tablet formulation of didanosine. Drug Dev. Ind. Pharm. 27 (2001) 129-136
2. Bonacucina G., Martelli S., and Palmieri G.F. Rheological, mucoadhesive and release properties of Carbopol gels in hydrophilic cosolvents. Int. J. Pharm. 282 (2004) 115-130
3. Chavasit V., Kienzle-Sterzer C., and Torres J.A. Formation and characterization of an insoluble polyelectrolyte complex: chitosan-polyacrylic acid. Polym. Bull. 19 (1988) 223-230
4. Chavasit V., and Torres J.A. Chitosan-poly(acrylic acid): mechanism of complex formation and potential industrial applications. Biotechnol. Prog. 6 (1990) 2-6
5. Cho S.-M., and Choi H.-K. Preparation of mucoadhesive chitosan-poly(acrylic acid) microspheres by interpolymer complexation and solvent evaporation method II. Arch. Pharm. Res. 28 (2005) 612-618
6. Cho S.-M., and Choi H.-K. Preparation of mucoadhesive chitosan-poly(acrylic acid) microspheres by interpolymer complexation and solvent evaporation method I. J. Kor. Pharm. Sci. 35 (2005) 95-99
7. de la Torre P.M., Enobakhare Y., Torrado G., and Torrado S. Release of amoxicillin from polyionic complexes of chitosan and poly(acrylic acid). Study of polymer/polymer and polymer/drug interactions within the network structure. Biomaterials 24 (2003) 1499-1506
8. ® compacts. Int. J. Pharm. 274 (2004) 233-243
9. Koleng J.J., and McGinity J.W. Carbomer. In: Kibbe A.H. (Ed). Handbook of Pharmaceutical Excipients. 3rd ed. (2000), Pharmaceutical Press, London, UK 79-82
10. Kranz H., Guthmann C., Wagner T., Lipp R., and Reiinhard J. Development of a single unit extended release formulation for ZK 811752, a weakly basic drug. Eur. J. Pharm. Sci. 26 (2005) 47-53
11. Lee I., and Peppas N.A. Prediction of polymer dissolution in swellable controlled-release systems. J. Control. Release 6 (1987) 207-215
12. Meshali M.M., El-Sayed G.M., El-Said Y., and Abd El-Aleem H.M. Preparation and evaluation of theophylline sustained release tablets. Drug Dev. Ind. Pharm. 22 (1996) 373-376
13. Mi F.-L., Shyu S.-S., Kuan C.-Y., Lee S.-T., Lu K.-T., and Jang S.-F. Chitosan-polyelectrolyte complexation for the preparation of gel beads and controlled release of anticancer drug. I. Effect of phosphorous polyelectrolyte complex and enzymatic hydrolysis of polymer. J. Appl. Polym. Sci. 74 (1999) 1868-1879
14. Nellore R.V., Rekhi G.S., Hussain A.S., Tillman L.G., and Augsburger L.L. Development of metoprolol tartrate extended-release matrix tablet formulations for regulatory policy consideration. J. Control. Release 50 (1998) 247-256
15. Neto C.G.T., Giacometti J.A., Job A.E., Ferreira F.C., Fonseca J.L.C., and Pereira M.R. Thermal analysis of chitosan based networks. Carbohyd. Polym. 62 (2005) 97-103
16. Nunthanid J., Laungtna-anan M., Sriamornsak P., Limmatvaprirat S., Puttipipatkhachorn S., Lim L.Y., and Khor E. Characterization of chitosan acetate as a binder for sustained release tablet. J. Control. Release 99 (2004) 15-26
17. Peppas N.A., and Sahlin J.J. A simple equation for the description of solute release. III. Coupling of diffusion and relaxation. Int. J. Pharm. 57 (1989) 169-172
18. Pretsch E., Buhlmann P., and Affolter C. Structure Determination of Organic Compounds: Tables of Spectral Data. 3rd ed. (2000), Springer, New York
19. Ritger P.L., and Peppas N.A. A simple equation for description of solute release. I. Fickian and non-fickian release from non-swellable devices in the form of slabs, sphere, cylinders or discs. J. Control. Release 5 (1987) 23-36
20. Shieh J.-J., and Huang R.Y.M. Pervaporation with chitosan membranes. II. Blend membranes of chitosan and polyacrylic acid and comparison of homogeneous and composite membrane based on polyelectrolyte complexes of chitosan and polyacrylic acid for the separation of ethanol-water mixtures. J. Membr. Sci. 127 (1997) 185-202
21. Singlga M., Chawla A., and Singh A. Potential applications of Carbomer in oral mucoadhesive controlled drug delivery system: a review. Drug Dev. Ind. Pharm. 26 (2000) 913-924
22. Tien C.L., Lacrix M., Ispas-Szabo P., and Mateescu M.-A. N-acylated chitosan: hydrophobic matrices for controlled drug release. J. Control. Release 93 (2003) 1-13
23. Vendruscolo C.W., Andreazza I.F., Ganter J.L.M.S., Ferrero C., and Bresolin T.M.B. Xanthan and galactomannan (from M. scabrella) matrix tablets for oral controlled delivery of theophylline. Int. J. Pharm. 296 (2005) 1-11
24. Wang H., Li W., Lu Y., and Wang Z. Studies on chitosan and poly (acrylic acid) interpolymer complex. I. Preparation, structure, pH-sensitivity, and salt sensitivity of complex-forming poly (acrylic acid): chitosan semi-interpenetrating polymer network. J. Appl. Polym. Sci. 65 (1997) 1445-1450
25. Zhong Z., and Guo Q. Interpolymer complexes and miscible blends of poly(N-vinyl-2-pyrrolidone) with novolac resin and the effect of crosslinking on related behaviour. Polym. Int. 41 (1996) 315-322