Preparation of rapidly disintegrating tablets containing itraconazole solid dispersions

Chemical and Pharmaceutical Bulletin

Volumn 55, Issue 11, 2007, Pages 1557-1562

  Oshima, Takao ^a   Sonoda, Ryoichi ^a   Ohkuma, Moriyuki ^a   Sunada, Hisakazu ^b  

^a KAKEN PHARMACEUTICAL CO LTD   (Japan)

^b MEIJO UNIVERSITY   (Japan)

Author keywords

Enteric polymer; Rapidly disintegrating tablet; Solid dispersion; Surface modifying

Indexed keywords

DISINTEGRATING AGENT; HYDROXYPROPYLMETHYLCELLULOSE PHTHALATE; ITRACONAZOLE; POLYMER; SILICIC ACID;

ARTICLE; DISPERSION; DRUG COATING; DRUG FORMULATION; DRUG GRANULATION; DRUG SOLUBILITY; DRUG SYNTHESIS; FLOW MEASUREMENT; TABLET DISINTEGRATION; TABLET HARDNESS; TABLET MACHINE;

ANTIFUNGAL AGENTS; CHEMISTRY, PHARMACEUTICAL; DITERPENES; DRUG STABILITY; EXCIPIENTS; ITRACONAZOLE; METHYLCELLULOSE; PARTICLE SIZE; SOLUBILITY; TABLETS, ENTERIC-COATED; TEMPERATURE; WATER;

EID: 36248942916     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.55.1557     Document Type: Article

References (26)

1. Japanese Package Insert of ITRIZOLE® Capsule 50 (14th), Janssen Pharmaceutical K.K., 2006.
2. Niewerth M., Korting H. C., Drugs, 58, 283-296 (1999).
3. Sato T., Koseki S., Takahashi S., Maie O., Mycoses, 33, 455-463 (1990).
4. Okuda C., Ito M., Jpn. J. Dermatol., 108, 733-738 (1998).
5. Willemsen M., De Doncker P., Willems J., Woestenborghs R., Van de Velde V., Heykants J., Van Cutsem J., Cauwenbergh G., Roseeuw D., J. Am. Acad. Dermatol., 26, 731-735 (1992).
6. Verreck G., Six K., Van den Mooter G., Baert L., Peeters J., Brewster M. E., Int. J. Pharm., 30, 165-174 (2003).
7. Baert L., Verreck G., Thone D., WO Patent 9744014 (1997).
8. Baert L., Peeters J., Verreck G., WO Patent 9701839 (1997).
9. Cha B. J., Oh J. G., Kim S. E., WO Patent 9857967 (1998).
10. Kwon J. W., Kim J. H., Wang H. S., Jang S. W., Bae W. T., WO Patent 200141765 (2001).
11. Senda S., Maeyama S., Jpn. Patent P2004-2245A (2004).
12. Ohara T., Kimura A., Jpn. Patent P2004-10575A (2004).
13. Van Peer A., Woestenborghs R., Heykants J., Gasparini R., Gauwenbergh G., Eur. J. Clin. Pharmacol., 36, 423-426 (1989).
14. Lange D., Pavao J. H., Wu J., Klausner M., J. Clin. Pharmacol., 37, 535-540 (1997).
15. Schmidt L. E., Dalhoff K., Drugs, 62, 1481-1502 (2002).
16. Fujishima I., Kurata N., "Simple Suspension Method, Naihukuyaku no Keikan Touyo Handbook," 2nd, Jiho, Tokyo. 2003.
17. Oshima T., Sonoda R., Ohkuma M., Sunada H., J. Pharm. Sci. Technol. Jpn., 67, 356-364 (2007).
18. Kato Y., Matsumoto K., Ohkuma M., Sunada H., J. Pharm. Sci. Technol. Jpn., 61, 109-118 (2001).
19. Kato Y., Matsumoto K., Ohkuma M., Sunada H., J. Pharm. Sci. Technol. Jpn., 62, 87-94 (2002).
20. "Guidelines for Bioequivalence Studies of Generic Products," Pharmaceutical and Medical Safety Bureau, Ministry of Health and Welfare, Notification No. 1124004, 2007.
21. Washburn E. W., Phys. Rev., 17, 273-281 (1921).
22. Oshima T., Sonoda R., Ohkuma M., Jpn. Patent P2006-143683A (2006).
23. Kato Y., Ohkuma M., Shimada Y., Sunada H., J. Drug Del. Sci. Tech., 15, 217-221 (2005).
24. Zhang G. G., Law D., Schmitt E. A., Qiu Y., Adv. Drug Deliv. Rev., 56, 371-390 (2004).
25. Nogami H., Nagai T., Fukuoka E., Yotusyanagi T., Chem. Pharm. Bull., 17, 23-31 (1969).
26. Zhao N., Augsburger L. L., AAPS Pharm. Sci. Tech., 17, 634-640 (2005).