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Volumn 42, Issue 10, 2007, Pages 601-608

Maraviroc: The first CCR5 antagonist for the treatment of HIV

Author keywords

[No Author keywords available]

Indexed keywords

ANTIRETROVIRUS AGENT; ATAZANAVIR; CHEMOKINE RECEPTOR CCR5; CHEMOKINE RECEPTOR CCR5 ANTAGONIST; CHEMOKINE RECEPTOR CXCR4; CLARITHROMYCIN; DELAVIRDINE; EFAVIRENZ; ENZYME INHIBITOR; ETHINYLESTRADIOL; ITRACONAZOLE; KETOCONAZOLE; LAMIVUDINE PLUS ZIDOVUDINE; LEVONORGESTREL; MARAVIROC; MIDAZOLAM; NEVIRAPINE; PLACEBO; RIFAMPICIN; RITONAVIR; SAQUINAVIR; TENOFOVIR; TIPRANAVIR;

EID: 35649011406     PISSN: 1082801X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review
Times cited : (3)

References (39)
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    • An investigation of the effects of tenofovir on the pharmacokinetics of the novel CCR5 inhibitor UK-427,857
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  • 33
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    • A study to investigate the combined co-administration of P450 CYP3A4 inhibitors and inducers on the pharmacokinetics of the novel CCR5 inhibitor UK-427,857
    • Presented at: November 14-17, Glasgow, UK. Abstract P284
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    • (2004) Seventh International Congress on Drug Therapy in HIV Infection
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  • 34
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    • An investigation of the effects of atazanavir and ritonavir boosted atazanavir on the pharmacokinetics of the novel CCR5 inhibitor UK-427,857
    • Presented at: November 14-17, Glasgow, UK. Abstract P283
    • Muirhead G, Abel S, Russell D, et al. An investigation of the effects of atazanavir and ritonavir boosted atazanavir on the pharmacokinetics of the novel CCR5 inhibitor UK-427,857. Presented at: Seventh International Congress on Drug Therapy in HIV Infection; November 14-17, 2004; Glasgow, UK. Abstract P283.
    • (2004) Seventh International Congress on Drug Therapy in HIV Infection
    • Muirhead, G.1    Abel, S.2    Russell, D.3
  • 35
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    • Effect of boosted tipranavir on the pharmacokinetics of maraviroc (UK 427,857) in healthy volunteers
    • November 17-20, Dublin, Ireland. Abstract LBPE4
    • Abel S, Taylor-Worth R, Ridgway C, Weissgerber G, Kraft M. Effect of boosted tipranavir on the pharmacokinetics of maraviroc (UK 427,857) in healthy volunteers. Poster presented at: 10th European AIDS Conference/EACS; November 17-20, 2005; Dublin, Ireland. Abstract LBPE4.3/15.
    • (2005) Poster presented at: 10th European AIDS Conference/EACS , pp. 3-15
    • Abel, S.1    Taylor-Worth, R.2    Ridgway, C.3    Weissgerber, G.4    Kraft, M.5
  • 36
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    • A novel probe drug interaction study to investigate the effect of selected ARV combinations on the pharmacokinetics of a single oral dose of maraviroc (UK-427,857) in HTV+ve subjects
    • April 28-30, Quebec, Canada. Poster 2.19
    • Muirhead G, Pozniak A, Boffito M, et al. A novel probe drug interaction study to investigate the effect of selected ARV combinations on the pharmacokinetics of a single oral dose of maraviroc (UK-427,857) in HTV+ve subjects. Poster presented at: 6th International Workshop on Clinical Pharmacology of HIV Therapy; April 28-30, 2005; Quebec, Canada. Poster 2.19.
    • (2005) Poster presented at: 6th International Workshop on Clinical Pharmacology of HIV Therapy
    • Muirhead, G.1    Pozniak, A.2    Boffito, M.3
  • 38
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    • Effect of UK-427,857, on the pharmacokinetics of oral contraceptive steroids, and the pharmacokinetics of UK-427,857 in healthy young women
    • Presented at: September 14-17, Chicago, IL. Abstract
    • Abel S, Whitlock L, Ridgway C, Saifulanwar A, Bakhtyari A, Russell D. Effect of UK-427,857, on the pharmacokinetics of oral contraceptive steroids, and the pharmacokinetics of UK-427,857 in healthy young women. Presented at: 43rd Interscience Conference on Antimicrobial Agents and Chemotherapy; September 14-17, 2003; Chicago, IL. Abstract A-1619.
    • (2003) 43rd Interscience Conference on Antimicrobial Agents and Chemotherapy
    • Abel, S.1    Whitlock, L.2    Ridgway, C.3    Saifulanwar, A.4    Bakhtyari, A.5    Russell, D.6


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