Overcoming inhibition

Nature Reviews Drug Discovery

Volumn 3, Issue 7, 2004, Pages 551-

  Jones, Daniel ^a  

^a NONE

Author keywords

[No Author keywords available]

Indexed keywords

4 (3 BROMOANILINO) 6,7 DIMETHOXYQUINAZOLINE; ADENOSINE TRIPHOSPHATE; EPIDERMAL GROWTH FACTOR RECEPTOR; GEFITINIB; IMATINIB; METHIONINE; OXINDOLE; PROTEIN KINASE; PROTEIN TYROSINE KINASE; PROTEIN TYROSINE KINASE INHIBITOR; THREONINE;

AMINO ACID SUBSTITUTION; BINDING SITE; CANCER RESEARCH; CARCINOGENESIS; DRUG SENSITIVITY; DRUG TARGETING; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME STRUCTURE; GENE MUTATION; HUMAN; MALIGNANT NEOPLASTIC DISEASE; MUTATIONAL ANALYSIS; NOTE; PRIORITY JOURNAL; PROTEIN TARGETING;

EID: 3543101369     PISSN: 14741776     EISSN: None     Source Type: Journal    
DOI: 10.1038/nrd1456     Document Type: Note

References (1)

1. Blencke, S. et al. Characterization of a conserved structural determinant controlling protein kinase sensitivity to selective inhibitors. Chem. Biol. 11, 691-701 (2004)