Geometry of GPPE binding to picrate and to the urokinase type plasminogen activator

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 22, 2007, Pages 6212-6215

  Zesławska, Ewa ^a   Stürzebecher, Jörg ^b   Oleksyn, Barbara J ^c  

^a PEDAGOGICAL UNIVERSITY   (Poland)

^b FRIEDRICH SCHILLER UNIVERSITY JENA   (Germany)

^c JAGIELLONIAN UNIVERSITY   (Poland)

Author keywords

Crystal structure; Inhibitor; Picrate; Urokinase; X ray diffraction

Indexed keywords

2 (4 GUANIDYNEPHENYL) 1 PHENYLETHANONE; ANTINEOPLASTIC AGENT; BENZENE DERIVATIVE; GUANIDINE DERIVATIVE; PICRIC ACID; UNCLASSIFIED DRUG; UROKINASE RECEPTOR;

ARTICLE; COMPLEX FORMATION; CRYSTAL STRUCTURE; DRUG CONFORMATION; DRUG RECEPTOR BINDING; DRUG TARGETING; GEOMETRY; HYDROGEN BOND; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION;

ANIONS; BINDING SITES; CRYSTALLOGRAPHY, X-RAY; GUANIDINES; HYDROGEN BONDING; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PICRATES; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; URINARY PLASMINOGEN ACTIVATOR;

EID: 35148894035     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.09.020     Document Type: Article

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