Synthesis and structure-activity relationship of 7-(substituted)-aminomethyl-4-quinolone-3-carboxylic acid derivatives

Bioorganic and Medicinal Chemistry

Volumn 15, Issue 23, 2007, Pages 7274-7280

  Zhang, Zhenfa ^a,b   Yu, Aizhen ^b   Zhou, Weicheng ^b  

^a University of Kentucky   (United States)

^b Shanghai Institute of Pharmaceutical Industry   (China)

Author keywords

Antibacterial agent; Fluoroquinolones; Gram positive bacteria

Indexed keywords

ANTIINFECTIVE AGENT; CARBOXYLIC ACID DERIVATIVE; PAZUFLOXACIN; VANCOMYCIN;

ANTIBACTERIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ANTI-BACTERIAL AGENTS; CARBOXYLIC ACIDS; DRUG DESIGN; KLEBSIELLA PNEUMONIAE; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; QUINOLONES; SALMONELLA; SHIGELLA BOYDII; STAPHYLOCOCCUS AUREUS; STEREOISOMERISM; STREPTOCOCCUS; STRUCTURE-ACTIVITY RELATIONSHIP;

NEGIBACTERIA; POSIBACTERIA;

EID: 35148890408     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2007.08.031     Document Type: Article

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