Virtual screening application of a model of full-length HIV-1 integrase complexed with viral DNA

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 19, 2007, Pages 5361-5365

  Liao, Chenzhong ^a   Karki, Rajeshri G ^a   Marchand, Christophe ^b   Pommier, Yves ^b   Nicklaus, Marc C ^a  

^a NATIONAL CANCER INSTITUTE   (United States)

^b NATIONAL CANCER INSTITUTE   (United States)

Author keywords

Computer aided drug design; Drug discovery; HIV 1 integrase strand transfer inhibitors; Virtual screening

Indexed keywords

INTEGRASE INHIBITOR; VIRUS DNA;

ARTICLE; CONTROLLED STUDY; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS 1; VIRUS MORPHOLOGY; WILD TYPE;

CATALYSIS; DNA, VIRAL; DRUG EVALUATION, PRECLINICAL; HIV INTEGRASE; HIV INTEGRASE INHIBITORS; HIV-1; HUMANS; MODELS, MOLECULAR; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 34548609774     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.08.011     Document Type: Article

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