Towards stereoselective radiosynthesis of α-[11C]methyl- substituted aromatic α-amino acids - A challenge of creation of quaternary asymmetric centre in a very short time

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 50, Issue 5-6, 2007, Pages 370-374

  Popkov, Alexander ^a,e   Nádvorník, Milan ^b   Kružberská, Pavla ^c   Lyčka, Antonín ^d   Lehel, Szabolcs ^e   Gillings, Nicholas ^e  

^a UNIVERSITY OF SOUTH BOHEMIA   (Czech Republic)

^b UNIVERSITY OF PARDUBICE   (Czech Republic)

^c INSTITUTE OF ENTOMOLOGY   (Czech Republic)

^d Vyzkumny ustav organickych syntez as   (Czech Republic)

^e Mental Health Services CPH   (Denmark)

Author keywords

Asymmetric synthesis; Carbon 11; Complexes; DOPA; Nickel; Tyrosine; 11C methylation; methyl amino acids

Indexed keywords

ALKYLATION; ENANTIOMERS; METHYLATION; NEURODEGENERATIVE DISEASES; NICKEL; POSITRON EMISSION TOMOGRAPHY; SODIUM HYDROXIDE; SYNTHESIS (CHEMICAL);

AMINO-ACIDS; ASYMMETRIC SYNTHESIS; CARBON-11; COMPLEX; DIASTEREOMERIC; DOPA; RADIOCHEMICAL YIELD; TYROSINE; [ 11C]METHYLATION; Α-METHYL AMINO ACID;

AMINO ACIDS;

1,3 DIMETHYLIMIDAZOLIDIN 2 ONE; ALPHA AMINO ACID C 11; METHYLDOPA C 11; METIROSINE C 11; RADIOPHARMACEUTICAL AGENT; SODIUM HYDROXIDE; UNCLASSIFIED DRUG;

CONFERENCE PAPER; DRUG STRUCTURE; DRUG SYNTHESIS; METHYLATION; POSITRON EMISSION TOMOGRAPHY; STEREOCHEMISTRY;

EID: 34548147019     PISSN: 03624803     EISSN: 10991344     Source Type: Journal    
DOI: 10.1002/jlcr.1268     Document Type: Conference Paper

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