Quantitative structure activity relationship studies of sulfamide derivatives as carbonic Anhydrase inhibitor: As antiglaucoma agents

Medicinal Chemistry

Volumn 3, Issue 4, 2007, Pages 379-386

  Kumar, Surendra ^a   Singh, Vineet ^b   Tiwari, Meena ^b  

^a Northern India Engineering College   (India)

^b SHRI G S INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

Anticancer drags; Antiviral drugs; Austin model 1; Carbonic anhydrase enzyme; Carbonic anhydrase inhibitors; Highest occupied molecular orbital; QSAR; Sulfamide derivative

Indexed keywords

ACETAZOLAMIDE; ANTIGLAUCOMA AGENT; BRINZOLAMIDE; CARBONATE DEHYDRATASE I; CARBONATE DEHYDRATASE II; CARBONATE DEHYDRATASE INHIBITOR; DICLOFENAMIDE; DORZOLAMIDE; ETHOXZOLAMIDE; METHAZOLAMIDE; SULFAMIDE DERIVATIVE;

ARTICLE; BOOTSTRAPPING; CALCULATION; CORRELATION COEFFICIENT; DEPENDENT VARIABLE; DRUG POTENCY; DRUG PROTEIN BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; ENZYME INHIBITION; GLAUCOMA; LINEAR REGRESSION ANALYSIS; PARAMETRIC TEST; PHYSICAL CHEMISTRY; PREDICTION; PRIORITY JOURNAL; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STATISTICAL SIGNIFICANCE; VALIDATION STUDY;

CARBONIC ANHYDRASE I; CARBONIC ANHYDRASE II; CARBONIC ANHYDRASE INHIBITORS; GLAUCOMA; HUMANS; MOLECULAR STRUCTURE; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 34447576540     PISSN: 15734064     EISSN: None     Source Type: Journal    
DOI: 10.2174/157340607781024447     Document Type: Article

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