Selective inhibition of the collagenase activity of cathepsin K

Journal of Biological Chemistry

Volumn 282, Issue 22, 2007, Pages 16492-16501

  Selent, Jana ^a   Kaleta, Jadwiga ^a   Li, Zhenqiang ^b   Lalmanach, Gilles ^c   Brömme, Dieter ^a  

^a UNIVERSITY OF BRITISH COLUMBIA   (Canada)

^b BRISTOL MYERS SQUIBB   (United States)

^c INSERM   (France)

Author keywords

[No Author keywords available]

Indexed keywords

COLLAGENASE ACTIVITY; NEGATIVE CHARGES;

BONE; CATALYST ACTIVITY; COLLAGEN; DEGRADATION;

ENZYME ACTIVITY;

AMINE; CATHEPSIN; CATHEPSIN K; CHONDROITIN 4 SULFATE; COLLAGENASE; CYANOGEN BROMIDE; FLUORESCEINAMINE; GLUTAMIC ACID; OLIGONUCLEOTIDE; POLYASPARTIC ACID; POLYGLUTAMIC ACID; POLYLYSINE; PROTEINASE; UNCLASSIFIED DRUG; CHONDROITIN SULFATE; COLLAGEN; MULTIPROTEIN COMPLEX;

ARTICLE; CATALYSIS; COLLAGEN DEGRADATION; CONTROLLED STUDY; DRUG MECHANISM; ENZYME ACTIVITY; ENZYME DEGRADATION; ENZYME INHIBITION; HUMAN; PRIORITY JOURNAL; PROTEIN DEGRADATION; CHEMISTRY; DRUG ANTAGONISM;

CATHEPSINS; CHONDROITIN SULFATES; COLLAGEN; COLLAGENASES; HUMANS; MULTIPROTEIN COMPLEXES; OLIGONUCLEOTIDES; POLYGLUTAMIC ACID;

EID: 34447509225     PISSN: 00219258     EISSN: 1083351X     Source Type: Journal    
DOI: 10.1074/jbc.M700242200     Document Type: Article

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