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Volumn 22, Issue 3, 2007, Pages 374-381

Five stabilized 111in-labeled neurotensin analogs in nude mice bearing HT29 tumors

Author keywords

111In labeled neurotensin analogs; Biodistribution; Exocrine pancreatic cancer; HT29 tumors; Serum stability

Indexed keywords

ARGININE; INDIUM 111; LYSINE; NEUROTENSIN; NEUROTENSIN RECEPTOR; PENTETATE INDIUM IN 111; PENTETREOTIDE; DRUG DERIVATIVE; INDIUM; OLIGOPEPTIDE; PENTETIC ACID;

EID: 34447503736     PISSN: 10849785     EISSN: None     Source Type: Journal    
DOI: 10.1089/cbr.2007.369.a     Document Type: Article
Times cited : (3)

References (32)
  • 2
    • 0023872949 scopus 로고
    • Pancreatic cancer: The greatest oncological challenge
    • Williamson RC. Pancreatic cancer: The greatest oncological challenge. Br Med J (Clin Res Ed) 1988;296: 445.
    • (1988) Br Med J (Clin Res Ed) , vol.296 , pp. 445
    • Williamson, R.C.1
  • 3
    • 0031911012 scopus 로고    scopus 로고
    • Epidemiology of and risk factors for pancreatic cancer
    • Gold EB, Goldin SB. Epidemiology of and risk factors for pancreatic cancer. Surg Oncol Clin N Am 1998;7:67.
    • (1998) Surg Oncol Clin N Am , vol.7 , pp. 67
    • Gold, E.B.1    Goldin, S.B.2
  • 4
    • 0018938939 scopus 로고
    • Report on a patient with watery diarrhoea syndrome caused by a pancreatic tumour containing neurotensin, enkephalin, and calcitonin
    • Gutniak M, Rosenqvist U, Grimelius L, et al. Report on a patient with watery diarrhoea syndrome caused by a pancreatic tumour containing neurotensin, enkephalin, and calcitonin. Acta Med Scand 1980;208:95.
    • (1980) Acta Med Scand , vol.208 , pp. 95
    • Gutniak, M.1    Rosenqvist, U.2    Grimelius, L.3
  • 5
    • 0034082312 scopus 로고    scopus 로고
    • Gut peptide receptor expression in human pancreatic cancers
    • Ehlers RA, Kim S, Zhang Y, et al. Gut peptide receptor expression in human pancreatic cancers. Ann Surg 2000;231:838.
    • (2000) Ann Surg , vol.231 , pp. 838
    • Ehlers, R.A.1    Kim, S.2    Zhang, Y.3
  • 6
    • 0031949569 scopus 로고    scopus 로고
    • Neurotensin receptors: A new marker for human ductal pancreatic adenocarcinoma
    • Reubi JC, Waser B, Friess H, et al. Neurotensin receptors: A new marker for human ductal pancreatic adenocarcinoma. Gut 1998;42:546.
    • (1998) Gut , vol.42 , pp. 546
    • Reubi, J.C.1    Waser, B.2    Friess, H.3
  • 7
    • 0032975129 scopus 로고    scopus 로고
    • Neurotensin receptors in human neoplasms: High incidence in Ewing's sarcomas
    • Reubi JC, Waser B, Schaer JC, et al. Neurotensin receptors in human neoplasms: High incidence in Ewing's sarcomas. Int J Cancer 1999;82:213.
    • (1999) Int J Cancer , vol.82 , pp. 213
    • Reubi, J.C.1    Waser, B.2    Schaer, J.C.3
  • 8
    • 0642310760 scopus 로고    scopus 로고
    • 99mTc-NT-XI, evaluated in ductal pancreatic adenocarcinoma patients
    • 99mTc-NT-XI, evaluated in ductal pancreatic adenocarcinoma patients. J Nucl Med 2003; 44:1649.
    • (2003) J Nucl Med , vol.44 , pp. 1649
    • Buchegger, F.1    Bonvin, F.2    Kosinski, M.3
  • 10
    • 0027207735 scopus 로고
    • Neurotensin regulates growth of human pancreatic cancer
    • Ishizuka J, Townsend CM, Jr, Thompson JC. Neurotensin regulates growth of human pancreatic cancer. Ann Surg 1993;217:439.
    • (1993) Ann Surg , vol.217 , pp. 439
    • Ishizuka, J.1    Townsend Jr, C.M.2    Thompson, J.C.3
  • 11
    • 0033956470 scopus 로고    scopus 로고
    • Neurotensin receptor-1 mRNA analysis in normal pancreas and pancreatic disease
    • Wang L, Friess H, Zhu Z, et al. Neurotensin receptor-1 mRNA analysis in normal pancreas and pancreatic disease. Clin Cancer Res 2000;6:566.
    • (2000) Clin Cancer Res , vol.6 , pp. 566
    • Wang, L.1    Friess, H.2    Zhu, Z.3
  • 12
    • 0027074957 scopus 로고
    • Biosynthesis, maturation, release, and degradation of neurotensin and neuromedin N
    • Kitabgi P, De Nadai F, Rovere C, et al. Biosynthesis, maturation, release, and degradation of neurotensin and neuromedin N. Ann N Y Acad Sci 1992;668:30.
    • (1992) Ann N Y Acad Sci , vol.668 , pp. 30
    • Kitabgi, P.1    De Nadai, F.2    Rovere, C.3
  • 13
    • 33646546315 scopus 로고    scopus 로고
    • 99mTc-labeled neurotensin peptide 8-13
    • 99mTc-labeled neurotensin peptide 8-13. Nucl Med Biol 2006;33:505.
    • (2006) Nucl Med Biol , vol.33 , pp. 505
    • Zhang, K.1    An, R.2    Gao, Z.3
  • 15
    • 33644854930 scopus 로고    scopus 로고
    • 99mTc-labeled neurotensin analogues with optimized biodistribution properties
    • 99mTc-labeled neurotensin analogues with optimized biodistribution properties. J Med Chem 2006;49:1833.
    • (2006) J Med Chem , vol.49 , pp. 1833
    • Maes, V.1    Garcia-Garayoa, E.2    Blauenstein, P.3
  • 16
    • 33646557942 scopus 로고    scopus 로고
    • Double-stabilized neurotensin analogues as potential radiopharmaceuticals for NTR-positive tumors
    • Garcia-Garayoa E, Maes V, Blauenstein P, et al. Double-stabilized neurotensin analogues as potential radiopharmaceuticals for NTR-positive tumors. Nucl Med Biol 2006;33:495.
    • (2006) Nucl Med Biol , vol.33 , pp. 495
    • Garcia-Garayoa, E.1    Maes, V.2    Blauenstein, P.3
  • 17
    • 0035138361 scopus 로고    scopus 로고
    • In vitro and in vivo evaluation of new radiolabeled neurotensin(8-13) analogues with high affinity for NT1 receptors
    • Garcia-Garayoa E, Allemann-Tannahill L, Blauenstein P, et al. In vitro and in vivo evaluation of new radiolabeled neurotensin(8-13) analogues with high affinity for NT1 receptors. Nucl Med Biol 2001;28:75.
    • (2001) Nucl Med Biol , vol.28 , pp. 75
    • Garcia-Garayoa, E.1    Allemann-Tannahill, L.2    Blauenstein, P.3
  • 18
    • 0026050226 scopus 로고
    • Reduced peptide bond pseudopeptide analogues of neurotensin: Binding and biological activities, and in vitro metabolic stability
    • Lugrin D, Vecchini F, Doulut S, et al. Reduced peptide bond pseudopeptide analogues of neurotensin: Binding and biological activities, and in vitro metabolic stability. Eur J Pharmacol 1991;205:191.
    • (1991) Eur J Pharmacol , vol.205 , pp. 191
    • Lugrin, D.1    Vecchini, F.2    Doulut, S.3
  • 19
    • 0043237915 scopus 로고    scopus 로고
    • 111In-labelled DTPA- and DOTA-conjugated neurotensin analogues for imaging and therapy of exocrine pancreatic cancer
    • 111In-labelled DTPA- and DOTA-conjugated neurotensin analogues for imaging and therapy of exocrine pancreatic cancer. Eur J Nucl Med Mol Imag 2003;30: 1134.
    • (2003) Eur J Nucl Med Mol Imag , vol.30 , pp. 1134
    • de Visser, M.1    Janssen, P.J.2    Srinivasan, A.3
  • 20
    • 0037700078 scopus 로고    scopus 로고
    • 177Lu at high specific activities. Eur J Nucl Med Mol Imag 2003;30:917.
    • 177Lu at high specific activities. Eur J Nucl Med Mol Imag 2003;30:917.
  • 21
    • 0035155042 scopus 로고    scopus 로고
    • Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals
    • Liu S, Edwards DS. Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals. Bioconjug Chem 2001;12:7.
    • (2001) Bioconjug Chem , vol.12 , pp. 7
    • Liu, S.1    Edwards, D.S.2
  • 24
    • 0034789911 scopus 로고    scopus 로고
    • Localization and characterization of neuropeptide receptors in human colon
    • Rettenbacher M, Reubi JC. Localization and characterization of neuropeptide receptors in human colon. Naunyn Schmiedebergs Arch Pharmacol 2001;364:291.
    • (2001) Naunyn Schmiedebergs Arch Pharmacol , vol.364 , pp. 291
    • Rettenbacher, M.1    Reubi, J.C.2
  • 25
    • 0036189966 scopus 로고    scopus 로고
    • Preclinical evaluation of a new, stabilized neurotensin (8-13) pseudopeptide radiolabeled with (99m)tc
    • Garcia-Garayoa E, Blauenstein P, Bruehlmeier M, et al. Preclinical evaluation of a new, stabilized neurotensin (8-13) pseudopeptide radiolabeled with (99m)tc. J Nucl Med 2002;43:374.
    • (2002) J Nucl Med , vol.43 , pp. 374
    • Garcia-Garayoa, E.1    Blauenstein, P.2    Bruehlmeier, M.3
  • 26
    • 0031475064 scopus 로고    scopus 로고
    • D-lysine reduction of indium-111 octreotide and yttrium-90 octreotide renal uptake
    • Bernard BF, Krenning EP, Breeman WA, et al. D-lysine reduction of indium-111 octreotide and yttrium-90 octreotide renal uptake. J Nucl Med 1997;38:1929.
    • (1997) J Nucl Med , vol.38 , pp. 1929
    • Bernard, B.F.1    Krenning, E.P.2    Breeman, W.A.3
  • 27
    • 0029738947 scopus 로고    scopus 로고
    • Inhibition of renal uptake of indium-111-DTPA-octreotide in vivo
    • de Jong M, Rolleman EJ, Bernard BF, et al. Inhibition of renal uptake of indium-111-DTPA-octreotide in vivo. J Nucl Med 1996;37:1388.
    • (1996) J Nucl Med , vol.37 , pp. 1388
    • de Jong, M.1    Rolleman, E.J.2    Bernard, B.F.3
  • 28
    • 9444265235 scopus 로고    scopus 로고
    • 99mTc-labeled anti-Tac disulfide-stabilized Fv fragment. Cancer Res 1996; 56:3788.
    • 99mTc-labeled anti-Tac disulfide-stabilized Fv fragment. Cancer Res 1996; 56:3788.
  • 29
    • 0030992080 scopus 로고    scopus 로고
    • Factors influencing the in vivo pharmacokinetics of peptides and antibody fragments: The pharmacokinetics of two PET-labeled low-molecular-weight proteins
    • Lang L, Jagoda E, Wu C, et al. Factors influencing the in vivo pharmacokinetics of peptides and antibody fragments: The pharmacokinetics of two PET-labeled low-molecular-weight proteins. Q J Nucl Med 1997;41:53.
    • (1997) Q J Nucl Med , vol.41 , pp. 53
    • Lang, L.1    Jagoda, E.2    Wu, C.3
  • 30
    • 0025939587 scopus 로고
    • Tolerance of normal tissue to therapeutic irradiation
    • Emami B, Lyman J, Brown A, et al. Tolerance of normal tissue to therapeutic irradiation. Int J Radiat Oncol Biol Phys 1991;21:109.
    • (1991) Int J Radiat Oncol Biol Phys , vol.21 , pp. 109
    • Emami, B.1    Lyman, J.2    Brown, A.3
  • 31
    • 0036148310 scopus 로고    scopus 로고
    • Biodistribution and catabolism of (18)F-labeled neurotensin (8-13) analogs
    • Bergmann R, Scheunemann M, Heichert C, et al. Biodistribution and catabolism of (18)F-labeled neurotensin (8-13) analogs. Nucl Med Biol 2002;29:61.
    • (2002) Nucl Med Biol , vol.29 , pp. 61
    • Bergmann, R.1    Scheunemann, M.2    Heichert, C.3
  • 32
    • 0036210651 scopus 로고    scopus 로고
    • Stabilization of neurotensin analogues: Effect on peptide catabolism, biodistribution and tumor binding
    • Bruehlmeier M, Garayoa EG, Blanc A, et al. Stabilization of neurotensin analogues: Effect on peptide catabolism, biodistribution and tumor binding. Nucl Med Biol 2002;29:321.
    • (2002) Nucl Med Biol , vol.29 , pp. 321
    • Bruehlmeier, M.1    Garayoa, E.G.2    Blanc, A.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.