Design space for a solventless photocurable pharmaceutical coating

Journal of Pharmaceutical Innovation

Volumn 1, Issue 1, 2006, Pages 44-53

  Bose, Sagarika ^a,b   Kelly, Brendan ^a,c   Bogner, Robin H ^a  

^a UNIVERSITY OF CONNECTICUT   (United States)

^b PFIZER INC   (United States)

^c MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

LACTOSE; POLYMER; SILOXANE;

ARTICLE; CONTROLLED STUDY; DRUG COATING; DRUG DOSAGE FORM; DRUG FORMULATION; FILM COATING; GOOD MANUFACTURING PRACTICE; INTERMETHOD COMPARISON; LIGHT EXPOSURE; LIGHT INTENSITY; LIQUID; PARTICLE SIZE; POWDER; PRIORITY JOURNAL; PROCESS DESIGN; PROCESS OPTIMIZATION; PROCESS TECHNOLOGY; SOLID STATE; SOLVENTLESS DRUG COATING;

EID: 34249102848     PISSN: 18725120     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF02784880     Document Type: Article

References (48)

1. Porter, S.C. (1982) The practical significance of the permeability and mechanical properties of polymer films used for the coating of pharmaceutical solid dosage forms. Int. J. Pharm. Technol. Prod. Manuf. 3, 21-25.
2. Banker, G.S. and Peck, G.E. (1981) The new, water-based colloidal dispersions. Pharm. Technol. 5, 55-61.
3. Porter, S.C. (1979) Aqueous film coating: an overview. Pharm. Technol. 3, 55-59.
4. Achanta, A.S. et al. (1997) Development of hot melt coating methods. Drug Dev. Ind. Pharm. 23, 441-449.
5. Joachim, J. and Cauture, E. (1996) A hot-melt coating agent for controlled-release. Pharmaceutical Manufacturing Review 8, 24-27.
6. Grosvenor, M.P. (1991) The physicomechanical properties of electrostatically deposited polymers for use in pharmaceutical powder coating, PhD thesis, Univ. Bath, Bath, UK.
7. Levinson, S.B. (1972) Electrocoat powder coat radiate. Which and why? II. Powder coat. J. Paint Technol. 44, 37-56.
8. Porter, S.C. Principles and application of dry powder deposition coating technology. AAPS Pharmaceutical Processing Conference, New Jersey, 2003.
9. Benoit, J.P. et al. Center de Microencapsulation. Method of coating particles. US Patent 6087003.
10. Thies, C. et al. (2003) A supercritical fluid-based coating technology 1: Process considerations. J. Microencapsul. 20, 87-96.
11. Ribeiro Dos Santos, I. et al. (2002) Microencapsulation of protein particles within lipids using a novel supercritical fluid process. Int. J. Pharm. 242, 69-78.
12. Wang, Y. et al. (2004) Polymer coating/encapsulation of nanoparticles using a supercritical anti-solvent process. The Journal of Supercritical Fluids 28, 85-99.
13. Yang, D.B. (1993) Kinetic studies of photopolymerization using real time FT-IR spectroscopy. J. Polym. Sci. Part A: Polym. Chem. 31, 199-208.
14. Yang, D.B. (1993) Direct kinetic measurements of vinyl polymerization on metal and silicon surfaces using real-time FT-IR spectroscopy. Appl. Spectrosc. 47, 1425-1429.
15. Roffey, C.G. (1982) Photopolymerization of Surface Coatings (1st edn). John Wiley and Sons.
16. Roffey, C.G. (1986) Ultraviolet curing for offset printing inks and varnishes. J. Oil Colour Chem. Assoc. 69, 288-296.
17. Roffey, C.G. (1998) Plastic cards and UV ink printing. Polymers Paint Colour J. 188, 30-34.
18. Kurze, U. Process and apparatus for UV-curing of plastics, Patent DE 4316862.
19. Tanoue, N. et al. (1998) The influence of ultraviolet radiation intensity on curing depth of photo-activated composite veneering materials. J. Oral Rehabil. 25, 770-775.
20. Lovell, L.G. et al. (2001) The effect of cure rate on the mechanical properties of dental resins. Dent. Mater. 17, 504-511.
21. Wilder, A.D. et al. (1983) Three-year clinical study of UV-cured composite resins in posterior teeth. J. Prosthet. Dent. 50, 26-30.
22. Wilder, A.D., Jr et al. (1999) Seventeen-year clinical study of ultraviolet-cured posterior composite Class I and II restorations. J. Esthet. Dent. 11, 135-142.
23. Burger, P. UV curing in medical applications. Medical Plastics, 2000, Collected Papers of the International Conference, 14th, Vienna, Austria (2000) 2.1-2.6.
24. Szycher, M. et al. Advanced UV-curable polyurethanes for wound dressings. Natl. SAMPE Symp. Exhib., [Proc.] 30 (Adv. Technol. Mater. Processes) (1985) 510-523.
25. Szycher, M. et al. Thermedics, Inc. (Woburn, MA). Drug dispensing wound dressing, US Patent 4614787.
26. Szycher, M. et al. (1986) Spandra: a sustained release battlefield wound dressing. J. Biomater. Appl. 1, 274-304.
27. Trotter, S. Beiersdorf AG (Hamburg, DE). Backing material for plasters and dressings, US Patent 6429154.
28. Lee, M.S. et al. Becton, Dickinson and Company (Franklin Lakes, NJ). Ultraviolet cured peelable film and method therefor, US Patent 5030665.
29. Pappas, S.P. (1985) UV curing by radical, cationic and concurrent radical-cationic polymerization. Radiat. Phys. Chem. 25, 633-641.
30. Kutal, C. et al. (1991) A novel strategy for photoinitiated anionic polymerization. Macromolecules 24, 6872-6873.
31. Otsubo, Y. et al. (1984) Rheological behavior of epoxy acrylate prepolymer during UV curing. J. Appl. Polym. Sci. 29, 4071-4080.
32. Decker, C. et al. (1980) Oxygen effect on UV curing and photodegradation of organic coatings. Org. Coat. Planst. Chem. 42, 710-715.
33. Wang, J.Z.Y. and Bogner, R.H. (1995) Solvent-free film coating using a novel photocurable polymer. Int. J. Pharm. 119, 81-89.
34. Savage, G.V. and Clevenger, J.M. Ciba-Geigy Corporation. Radiation cured drug release controlling membrane, US Patent 5532287.
35. Savage, G.V. and Clevenger, J.M. Ciba-Geigy Corporation. Method of using a radiation cured drug release controlling membrane, US Patent 5545442.
36. Keningley, S.T. et al. (1997) An investigation into the effects of binder viscosity on agglomeration behavior. Powder Technology 91, 95-103.
37. Rowe, R.C. (1989) Binder-substrate interactions in granulation; a theoretical approach based on surface free energy and polarity. Int. J. Pharm. 52, 149-154.
38. Hapgood, K.P. et al. (2002) Drop penetration into porous powder beds. J. Colloid Interface Sci. 253, 353-366.
39. Kennedy, J.P. and Niebergall, P.J. (1997) Preliminary assessment of an image analysis method for the evaluation of pharmaceutical coatings. Pharm. Dev. Technol. 2, 205-212.
40. Atai, M. et al. (2004) Physical and mechanical properties of an experimental dental composite based on a new monomer. Dent. Mater. 20, 663-668.
41. Tarumi, H. et al. (1999) Post-irradiation polymerization of composites containing bis-GMA and TEGDMA. Dent. Mater. 15, 238-242.
42. Imazato, S. et al. (1999) Water sorption, degree of conversion, and hydrophobicity of resins containing Bis-GMA and TEGDMA. Dent. Mater. 18, 124-132.
43. Kim, S. and Jang, J. (1996) The measurement of degree of conversion of BisGMA/silica composites by FTIR spectroscopy. Polymer Testing 15, 559-571.
44. Hussain Latiff, A. et al. (2005) Properties of eight methacrylated beta-cyclodextrin composite formulations. Dent. Mater. 21, 210-216.
45. Imazato, S. et al. (2001) Degree of conversion of composites measured by DTA and FTIR. Dent. Mater. 17, 178-183.
46. Lu, H. et al. (2004) Towards the elucidation of shrinkage stress development and relaxation in dental composites. Dent. Mater. 20, 979-986.
47. Mendes, L.C. et al. (2005) Determination of degree of conversion as function of depth of a photo-initiated dental restoration composite. Polymer Testing 24, 418-422.
48. Simons, S.J.R. and Fairbrother, R.J. (2000) Direct observations of liquid binder-particle interactions: the role of wetting behavior in agglomerate growth. Powder Technology 110, 44-58.