One-pot synthesis of substituted 2-aminobenzo[b]thiophenes

Journal of Organic Chemistry

Volumn 72, Issue 8, 2007, Pages 3122-3124

  Solovyev, Andrey Y ^a   Androsov, Dmitry A ^a   Neckers, Douglas C ^a  

^a BOWLING GREEN STATE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINOBENZOTHIOPHENES; SECONDARY AMINES; WILLGERODT KINDLER ROUTES;

AMINES; AMINO ACIDS; BENZENE; REACTION KINETICS; SUBSTITUTION REACTIONS; SYNTHESIS (CHEMICAL);

OLEFINS;

1 (2 CHLORO 5 NITROPHENYL)ETHANONE; 2 AMINOBENZO[B]THIOPHENE DERIVATIVE; AMINE; BENZENE DERIVATIVE; THIOPHENE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; ONE POT SYNTHESIS; REACTION ANALYSIS; SYNTHESIS;

EID: 34247193661     PISSN: 00223263     EISSN: None     Source Type: Journal    
DOI: 10.1021/jo062141a     Document Type: Article

References (16)

1. Grese, T. A.; Pennington, L. D.; Sluka, J. P.; Adrian, M. D.; Cole, H. W.; Fuson, T. R.; Magee, D. E.; Phillips, D. L.; Rowley, E. R.; Shetler, P. K.; Short, L. L.; Venugopalan, M.; Yang, N. N.; Sato, M.; Glasebrook, A. L.; Bryant, H. U. J. Med. Chem. 1998, 41, 1272-1283.
2. Grese, T. A.; Cho, S.; Finley, D. R.; Godfrey, A. G.; Jones, C. D.; Lugar, C. W.; Martin, M. J.; Matsumoto, K.; Pennington, L. D.; Winter, M. A.; Adrian, M. D.; Cole, H. W.; Magee, D. E.; Phillips, D. L.; Rowley, E. R.; Short, L. L.; Glasebrook, A. L.; Bryant, H. U. J. Med. Chem. 1997, 40, 146-167.
3. Lee, K. C.; Moon, B. C.; Lee, J. H.; Chung, K.-H.; Katzenellenbogen, J. A.; Chi, D. Y. Bioorg. Med. Chem. 2003, 11, 3649-3658.
4. Takeuchi, K.; Kohn, T. J.; Sall, D. J.; Denney, M. L.; McCowan, J. R.; Smith, G. F.; Gifford-Moore, D. S. Bioorg. Med. Chem. 1999, 9, 759-764.
5. Stacy, G. W.; Villaescusa, F. W.; Wollner, T. E. J. Org. Chem. 1965, 30, 4074-4078.
6. Grandclaudon, P.; Lablache-Combier, A. J. Org. Chem. 1978, 43, 4379-4381.
7. Brower, K. R.; Amstutz, E. D. J. Org. Chem. 1954, 19, 411-414.
8. Benincori, T.; Sannicolo, F. J. Org. Chem. 1988, 53, 1309-1312.
9. Zbruev, O. I.; Stiasni, N.; Kappe, C. O. J. Comb. Chem. 2003, 5, 145-148.
10. U.S. Patent 6.355,796 B1.
11. Schwenk, E.; Bloch, E. J. Am. Chem. Soc. 1942, 64, 3051-3052.
12. Klingele, M. H.; Brooker, S. Eur. J. Org. Chem. 2004, 3422-3434.
13. Poupaert, J. H.; Duarte, S.; Colacino, E.; Depreux, P.; McCurdy, C. M.; Lambert, D. L. Phosphorus, Sulfur Silicon Relat. Elem. 2004, 179, 1959-1973.
14. Aghapoor, K.; Darabi, H.-R.; Tabar-Heydar, K. Phosphorus, Sulfur Silicon Relat. Elem. 2002, 177, 1183-1187.
15. Aghapoor, K.; Darabi, H.-R.; Tabar-Heydar, K. Phosphorus, Sulfur Silicon Relat. Elem. 2002, 177, 1189-1192.
16. Schroth, W.; Andersch, J. Synthesis 1989, 202-204.