1,2,3-Triazolylalkylribitol derivatives as nucleoside hydrolase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 9, 2007, Pages 2523-2526

  Goeminne, A ^a   McNaughton, M ^a   Bal, G ^a   Surpateanu, G ^a   Van der Veken, P ^a   De Prol, S ^b,c   Versees W ^b,c   Steyaert, J ^b,c   Apers, S ^a   Haemers, A ^a   Augustyns, K ^a  

^a UNIVERSITY OF ANTWERP   (Belgium)

^b VRIJE UNIVERSITEIT BRUSSEL   (Belgium)

^c DEPARTMENT OF PLANT SYSTEMS BIOLOGY   (Belgium)

Author keywords

1,2,3 Triazolylalkylribitol; 1,3 Dipolar cycloaddition; Nucleoside hydrolase inhibitors

Indexed keywords

5 METHYL 4 PHENYL 1,2,3 TRIAZOLYLIMINORIBITOL DERIVATIVE; HYDROLASE INHIBITOR; IMMUCILLIN H; NUCLEOSIDE HYDROLASE INHIBITOR; RIBITOL DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS;

ANIMALS; CHEMISTRY, PHARMACEUTICAL; DRUG DESIGN; ENZYME INHIBITORS; KINETICS; MODELS, CHEMICAL; MOLECULAR CONFORMATION; N-GLYCOSYL HYDROLASES; RIBITOL; TRIAZOLES; TRYPANOSOMA BRUCEI BRUCEI;

EID: 33947723602     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.02.017     Document Type: Article

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