Distinct activity of peptide mimetic intracellular ligands (pepducins) for proteinase-activated receptor-1 in multiple cells/tissues

Annals of the New York Academy of Sciences

Volumn 1091, Issue , 2006, Pages 445-459

  Kubo, Satoko ^a   Ishiki, Tsuyoshi ^a   Doe, Ichiko ^a   Sekiguchi, Fumiko ^a   Nishikawa, Hiroyuki ^b   Kawai, Kenzo ^b   Matsui, Hirofumi ^c   Kawabata, Atsufumi ^a  

^a KINKI UNIVERSITY   (Japan)

^b Fuso Pharmaceutical Industries Ltd   (Japan)

^c UNIVERSITY OF TSUKUBA   (Japan)

Author keywords

Intracellular ligands; Palmitoylated peptide; Pepducin; Proteinase activated receptor 1 (PAR1); Thrombin

Indexed keywords

PEPDUCIN; PEPTIDE DERIVATIVE; PROTEIN INHIBITOR; PROTEINASE ACTIVATED RECEPTOR 1; UNCLASSIFIED DRUG; LIGAND; PEPTIDE;

ANIMAL CELL; ANIMAL EXPERIMENT; AORTA; CALCIUM MOBILIZATION; CONFERENCE PAPER; CONTROLLED STUDY; CYTOSOL; DESENSITIZATION; HUMAN; HUMAN CELL; LUNG ALVEOLUS EPITHELIUM; MALE; MOUSE; NONHUMAN; PALMITOYLATION; PROTEIN EXPRESSION; RAT; SMOOTH MUSCLE; SMOOTH MUSCLE FIBER; STOMACH EPITHELIUM; STOMACH MUCOSA; VASCULAR ENDOTHELIUM; VASODILATATION; AMINO ACID SEQUENCE; ANIMAL; ARTICLE; BIOMIMETICS; CELL LINE; CHEMISTRY; DRUG ANTAGONISM; INTRACELLULAR FLUID; METABOLISM; MOLECULAR GENETICS; MUSCLE RELAXATION; PHYSIOLOGY; PROTEIN BINDING; TUMOR CELL LINE; WISTAR RAT;

RATTUS;

AMINO ACID SEQUENCE; ANIMALS; BIOMIMETICS; CELL LINE; CELL LINE, TUMOR; HUMANS; INTRACELLULAR FLUID; LIGANDS; MALE; MICE; MOLECULAR SEQUENCE DATA; MUSCLE RELAXATION; PEPTIDES; PROTEIN BINDING; RATS; RATS, WISTAR; RECEPTOR, PAR-1;

EID: 33947600810     PISSN: 00778923     EISSN: 17496632     Source Type: Book Series    
DOI: 10.1196/annals.1378.087     Document Type: Conference Paper

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