Preparation, in vitro, preclinical and clinical evaluations of once daily sustained release tablets of aceclofenac

Archives of Pharmacal Research

Volumn 30, Issue 2, 2007, Pages 222-234

  Mutalik, S ^a   Naha, A ^a   Usha, A N ^a   Ranjith, A K ^a   Musmade, P ^a   Manoj, K ^a   Anju, P ^a   Prasanna, S ^b  

^a MANIPAL COLLEGE OF PHARMACEUTICAL SCIENCES   (India)

^b Exela Pharm Science Pvt Ltd   (India)

Author keywords

Aceclofenac; Analgesic; Anti inflammatory; Direct compression; Hydroxypropyl methylcellulose; Matrix tablets; Once daily; Pharmacokinetics; Sustained release; Toxicity

Indexed keywords

EID: 33947165208     PISSN: 02536269     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF02977698     Document Type: Article

References (22)

1. Alderman, D. A., A review of cellulose ethers in hydrophilic matrices for oral controlled dosage forms. Int. J. Pharm. Tech. Prod. Manuf., 3, 1-9 (1984).
2. Amaral, M. H., Lobo, J. M., and Ferreira, D. C., Effect of hydroxypropyl methylcellulose and hydrogenated castor oil on naproxen release from sustained-release tablets. AAPS. PharmSciTech., 2, article 6: 1-8, (2001).
3. Aulton, E. M., Pharmaceutics-The Science of Dosage Form Design. ELBS/ Churchill Livingstone, London, (1990).
4. British Pharmacopoeia. The Stationary office, MHRA, British Pharmacopoeial Commission office, Vol. 1, London, (2005).
5. Chien, Y. W., Regulatory considerations in controlled release medication, In Chien, Y. W. (Eds.). Novel Drug Delivery Systems. Marcel Dekker, New York, pp. 577-578, (1982).
6. Ford, J. L., Rubinstein, M. H., and Hogan, J. E., Formulation of sustained-release promethazine hydrochloride tablets using hydroxypropyl methylcellulose matrices. Int. J. Pharm., 24, 327-338 (1985).
7. Indian Pharmacopoeia, Ministry of Health and Family Welfare, Government of India, Controller of Publications, Vol. 2, Delhi, (1996).
8. rd ed., Churchill Livingstone, London, pp. 791-807, (2003).
9. Kuksal, A., Tiwary, A. K., Jain, N. K., and Jain, S., Formulation and In Vitro, In Vivo Evaluation of Extendedrelease Matrix Tablet of Zidovudine: Influence of Combination of Hydrophilic and Hydrophobic Matrix Formers. AAPS. PharmSciTech., 1, Article 1: 1-9, (2006).
10. Kulkarni, S.K., Handbook of experimental pharmacology, 2nd edn., Vallabh Prakashan, New Delhi, (1997).
11. Liebermann, H. A., Lachman, L., and Schwartz, J. B., Pharmaceutical Dosage Forms: Tablets, Vol. 2, Marcel Dekker, New York, pp. 201-243, (1990).
12. rd ed., Varghese Publishing House, New Delhi, pp. 442-454, (1991).
13. Mahaguna, V., Talbert, R. L., Peters, J. I., Adams, S., Reynolds, T. D., and Lam, F. Y. W., Influence of hydroxypropyl methylcellulose polymer on in vitro and in vivo performance of controlled release tablets containing alprazolam. Eur. J. Pharm. Biopharm., 56, 461-468, (2003).
14. Mutalik, S. and Hiremath, D., Formulation and evaluation of chitosan matrix tablets of nifedipine. The Eastern. Pharmacist., 10, 109-111, (2000).
15. Mutalik, S., Paridhavi, K., Rao, M., and Udupa, N., Analgesic and antipyretic effect of Solanum melongena. Indian J. Pharmacol., 32, 312-315 (2003a).
16. Mutalik, S., Sulochana, B., Chetana, M., Udupa, N., and Uma Devi, P., Preliminary studies on acute and subacute toxicity studies of an antidiabetic herbal formulation, Dianex. Indian J. Exptl. Biol., 4, 316-320 (2003b).
17. Mutalik, S. and Udupa, N., Formulation development, in vitro and in vivo evaluation of membrane controlled transdermal systems of glibenclamide. J. Pharm. Pharmaceut. Sci., 1, 26-38 (2005).
18. Nellore, R. V., Rekhi, G. S., Hussain, A. S., Tillman, L. G., and Augsburger, L. L., Development of metoprolol tartrate extended-release matrix tablet formulations for regulatory policy consideration. J. Controlled. Rel., 50, 247-256, (1998).
19. nd ed., Massachusetts, pp. 2-12, (1999).
20. Reddy, R., Mutalik, S., and Reddy, M. S., Once daily sustained release matrix tablets of nicorandil: Formulation and in vitro evaluation. AAPS. PharmSciTech., 4, Article 61: 1-9, (2003).
21. Terashita, K. and Imamura, K., Preparation of antipyretic analgesic by direct compression and its evaluation. Chem. Pharm. Bull., 12,1542-1549, (2002).
22. Vueba, M. L., Batista, D. C., Veiga, F., Sousa, J. J., and Pina, M. E., Influence of cellulose ether polymers on ketoprofen release from hydrophilic matrix tablets. Eur. J. Pharm. Biopharm., 1, 51-59 (2004).