메뉴 건너뛰기




Volumn 57, Issue 1, 2007, Pages 99-109

Liquisolid technique as a tool for enhancement of poorly water-soluble drugs and evaluation of their physicochemical properties

Author keywords

Aging; Dissolution rate; DSC; Indomethacin; Liquisolid compacts; XPD

Indexed keywords

INDOMETACIN; MACROGOL 400; MICROCRYSTALLINE CELLULOSE; POLYSORBATE 80; PROPYLENE GLYCOL; SILICON DIOXIDE;

EID: 33847617927     PISSN: 13300075     EISSN: None     Source Type: Journal    
DOI: 10.2478/v10007-007-0008-6     Document Type: Article
Times cited : (55)

References (21)
  • 1
    • 0035965506 scopus 로고    scopus 로고
    • Processing factors in development of solid solution formulation of itraconazole for enhancement of drug dissolution and bioavailability
    • S. G. Kapsi and J. W. Ayres, Processing factors in development of solid solution formulation of itraconazole for enhancement of drug dissolution and bioavailability, Int. J. Pharm. 229 (2001) 193-203.
    • (2001) Int. J. Pharm , vol.229 , pp. 193-203
    • Kapsi, S.G.1    Ayres, J.W.2
  • 2
    • 0014136951 scopus 로고
    • Deagglomeration behavior of relatively insoluble benzoic acid and its sodium salt
    • A. J. Aguiar, A. J. Zelmer and A. W. Kinkel, Deagglomeration behavior of relatively insoluble benzoic acid and its sodium salt, J. Pharm. Sc. 56 (1967) 1243-1252.
    • (1967) J. Pharm. Sc , vol.56 , pp. 1243-1252
    • Aguiar, A.J.1    Zelmer, A.J.2    Kinkel, A.W.3
  • 3
    • 0014318742 scopus 로고
    • Dissolution kinetics of drugs in human gastric juice; the role of surface tension
    • P. Finholt and S. Solvang, Dissolution kinetics of drugs in human gastric juice; the role of surface tension, J. Pharm. Sci. 57 (1968) 1322-1326.
    • (1968) J. Pharm. Sci , vol.57 , pp. 1322-1326
    • Finholt, P.1    Solvang, S.2
  • 4
    • 0014384257 scopus 로고
    • Interdependence of physiological surfactant and drug particle size on the dissolution behavior of water insoluble drugs
    • S. L. Lin, J. Menig and L. Lachman, Interdependence of physiological surfactant and drug particle size on the dissolution behavior of water insoluble drugs, J. Pharm. Sci. 57 (1968) 2143-2146.
    • (1968) J. Pharm. Sci , vol.57 , pp. 2143-2146
    • Lin, S.L.1    Menig, J.2    Lachman, L.3
  • 5
    • 0032543173 scopus 로고    scopus 로고
    • Enhancement of prednisolone dissolution properties using liquisolid compacts
    • S. Spireas and S. Sadu, Enhancement of prednisolone dissolution properties using liquisolid compacts, Int. J. Pharm. 166 (1998) 177-188.
    • (1998) Int. J. Pharm , vol.166 , pp. 177-188
    • Spireas, S.1    Sadu, S.2
  • 6
    • 0032109669 scopus 로고    scopus 로고
    • In vitro release evaluation of hydrocortisone liquisolid tablets
    • S. Spireas, S. Sadu and R. Grover, In vitro release evaluation of hydrocortisone liquisolid tablets, J. Pharm. Sci. 87 (1998) 867-872.
    • (1998) J. Pharm. Sci , vol.87 , pp. 867-872
    • Spireas, S.1    Sadu, S.2    Grover, R.3
  • 7
    • 0032968283 scopus 로고    scopus 로고
    • Effect of powder substrate on the dissolution properties of methchrothiazide liquisolid compacts
    • S. Spireas, T. Wang and R. Grover, Effect of powder substrate on the dissolution properties of methchrothiazide liquisolid compacts, Drug Dev. Ind. Pharm. 25 (1999) 163-168.
    • (1999) Drug Dev. Ind. Pharm , vol.25 , pp. 163-168
    • Spireas, S.1    Wang, T.2    Grover, R.3
  • 8
    • 0018761797 scopus 로고
    • Effect of amorphous silicon dioxide on drug dissolution
    • K. Y. Yang, R. Glemza and C. I. Jarowski, Effect of amorphous silicon dioxide on drug dissolution, J. Pharm. Sci. 68 (1979) 560-565.
    • (1979) J. Pharm. Sci , vol.68 , pp. 560-565
    • Yang, K.Y.1    Glemza, R.2    Jarowski, C.I.3
  • 9
    • 0021349430 scopus 로고
    • Dissolution rates of corticoid solutions dispersed on silicas
    • C. Liao and C. I. Jarowski, Dissolution rates of corticoid solutions dispersed on silicas, J. Pharm. Sci. 73 (1984) 401-403.
    • (1984) J. Pharm. Sci , vol.73 , pp. 401-403
    • Liao, C.1    Jarowski, C.I.2
  • 10
    • 27444438012 scopus 로고    scopus 로고
    • The effect of type and concentration of vehicles on the dissolution rate of a poorly soluble drug (indomethacin) from liquisolid compacts
    • A. Nokhodchi, Y. Javadzadeh, M. R. Siahi and M. Barzegar-Jalali, The effect of type and concentration of vehicles on the dissolution rate of a poorly soluble drug (indomethacin) from liquisolid compacts, J. Pharm. Pharm. Sci. 8 (2005) 18-25.
    • (2005) J. Pharm. Pharm. Sci , vol.8 , pp. 18-25
    • Nokhodchi, A.1    Javadzadeh, Y.2    Siahi, M.R.3    Barzegar-Jalali, M.4
  • 12
    • 0035806261 scopus 로고    scopus 로고
    • An alternative method to the evaluation of similarity factor in dissolution testing
    • P. Costa, An alternative method to the evaluation of similarity factor in dissolution testing, Int. J. Pharm. 220 (2001) 77-83.
    • (2001) Int. J. Pharm , vol.220 , pp. 77-83
    • Costa, P.1
  • 13
    • 0035073301 scopus 로고    scopus 로고
    • Modelling and comparison of dissolution profiles
    • P. Costa and J. M. S. Lobo, Modelling and comparison of dissolution profiles, Eur. J. Pharm. Sci. 13 (2001) 123-133.
    • (2001) Eur. J. Pharm. Sci , vol.13 , pp. 123-133
    • Costa, P.1    Lobo, J.M.S.2
  • 14
    • 0016422844 scopus 로고
    • Concept of dissolution efficiency
    • K. A. Khan, Concept of dissolution efficiency, J. Pharm. Pharmacol. 27 (1975) 48-49.
    • (1975) J. Pharm. Pharmacol , vol.27 , pp. 48-49
    • Khan, K.A.1
  • 16
    • 0022368809 scopus 로고
    • Physicochemical characterization of indomethacin polymorphs and transformation kinetics in ethanol
    • N. Kaneniwa, M. Otsuka and T. Hayashi, Physicochemical characterization of indomethacin polymorphs and transformation kinetics in ethanol, Chem. Pharm. Bull. 33 (1985) 3447-3455.
    • (1985) Chem. Pharm. Bull , vol.33 , pp. 3447-3455
    • Kaneniwa, N.1    Otsuka, M.2    Hayashi, T.3
  • 17
    • 0019119506 scopus 로고
    • Stability of several physical properties of amorphous and crystalline forms of indomethacin
    • H. Imaizumi, N. Nambu and T. Nagai, Stability of several physical properties of amorphous and crystalline forms of indomethacin, Chem. Pharm. Bull. 28 (1980) 2565-2569.
    • (1980) Chem. Pharm. Bull , vol.28 , pp. 2565-2569
    • Imaizumi, H.1    Nambu, N.2    Nagai, T.3
  • 18
    • 0016249928 scopus 로고
    • Polymorphism of indomethacin. New modifications, their melting behavior and solubility
    • L. Borka, Polymorphism of indomethacin. New modifications, their melting behavior and solubility, Acta Pharm. Suecica 11 (1974) 295-303.
    • (1974) Acta Pharm. Suecica , vol.11 , pp. 295-303
    • Borka, L.1
  • 19
    • 0034822729 scopus 로고    scopus 로고
    • Determination of indomethacin polymorphic contents by chemometric near-infrared spectroscopy and conventional powder X-ray diffractometry
    • M. Otsuka, F. Kato and Y. Matsuda, Determination of indomethacin polymorphic contents by chemometric near-infrared spectroscopy and conventional powder X-ray diffractometry, Analyst 126 (2001) 1578-1582.
    • (2001) Analyst , vol.126 , pp. 1578-1582
    • Otsuka, M.1    Kato, F.2    Matsuda, Y.3
  • 20
    • 0028597539 scopus 로고
    • Crystallization of indomethacin from the amorphous state below and above its glass transition temperature
    • M. Yoshioka, B.C. Hancock and G. Zografi, Crystallization of indomethacin from the amorphous state below and above its glass transition temperature, J. Pharm. Sci. 83 (1994) 1700-1705.
    • (1994) J. Pharm. Sci , vol.83 , pp. 1700-1705
    • Yoshioka, M.1    Hancock, B.C.2    Zografi, G.3
  • 21
    • 0020591926 scopus 로고
    • Stabilization of amorphous state of indomethacin by solid dispersions in polyvinylpyrolidone
    • H. Imaizumi, N. Nambu and T. Nagai, Stabilization of amorphous state of indomethacin by solid dispersions in polyvinylpyrolidone, Chem. Pharm. Bull. 31 (1983) 2510-2512.
    • (1983) Chem. Pharm. Bull , vol.31 , pp. 2510-2512
    • Imaizumi, H.1    Nambu, N.2    Nagai, T.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.