The channel-lining 6′ amino acid in the second membrane-spanning region of ionotropic GABA receptors has more profound effects on 4′-ethynyl-4-n-propylbicycloorthobenzoate binding than the 2′ amino acid

Invertebrate Neuroscience

Volumn 7, Issue 1, 2007, Pages 39-46

  Hisano, Kazutoshi ^a   Ozoe, Fumiyo ^a   Huang, Jia ^a   Kong, Xiangyu ^a   Ozoe, Yoshihisa ^a  

^a SHIMANE UNIVERSITY   (Japan)

Author keywords

Antagonist; Binding site; EBOB; GABA receptor; Housefly

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID A RECEPTOR BETA 3; AMINO ACID DERIVATIVE; BENZOIC ACID DERIVATIVE; MUTANT PROTEIN; OLIGOMER; RECEPTOR SUBUNIT; UNCLASSIFIED DRUG;

AMINO ACID SUBSTITUTION; BINDING KINETICS; BINDING SITE; CONFERENCE PAPER; GENETIC TRANSFECTION; INSECT CELL; MOLECULAR INTERACTION; MOLECULAR MODEL; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; RECEPTOR BINDING; RECEPTOR GENE; SEQUENCE HOMOLOGY;

AMINO ACID SUBSTITUTION; BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING SITES; DNA PRIMERS; HUMANS; INSECTICIDES; MODELS, MOLECULAR; MOLECULAR CONFORMATION; POLYMERASE CHAIN REACTION; PROTEIN CONFORMATION; RECEPTORS, GABA-A; STRUCTURE-ACTIVITY RELATIONSHIP; TRITIUM;

EID: 33847341155     PISSN: 13542516     EISSN: None     Source Type: Journal    
DOI: 10.1007/s10158-006-0035-x     Document Type: Conference Paper

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