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Volumn 1, Issue 12, 2006, Pages 1379-1390

Arylthiopyrrole (AThP) derivatives as non-nucleoside HIV-1 reverse transcriptase inhibitors: Synthesis, structure-activity relationships, and docking studies (Part 2)

(9) Lavecchia, Antonio b Costi, Roberta a Artico, Marino a Miele, Gaetano a Novellino, Ettore b Bergamini, Alberto c Crespan, Emmanuele d Maga, Giovanni d Di Santo, Roberto a

a SAPIENZA UNIVERSITY OF ROME (Italy)

b UNIVERSITY OF NAPLES FEDERICO II (Italy)

c UNIVERSITY OF ROME TOR VERGATA (Italy)

d CNR (Italy)

Author keywords

AIDS; Antiviral agents; Arylthiopyrroles; HIV; NNRTI

Indexed keywords

LIGAND; PYRROLE DERIVATIVE; RNA DIRECTED DNA POLYMERASE; RNA DIRECTED DNA POLYMERASE INHIBITOR;

ARTICLE; BINDING SITE; CELL LINE; CHEMICAL STRUCTURE; CHEMISTRY; COMPUTER SIMULATION; DRUG ANTAGONISM; DRUG DESIGN; DRUG EFFECT; HUMAN; HUMAN IMMUNODEFICIENCY VIRUS 1; MICROBIOLOGICAL EXAMINATION; STEREOISOMERISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS; X RAY CRYSTALLOGRAPHY;

BINDING SITES; CELL LINE; COMPUTER SIMULATION; CRYSTALLOGRAPHY, X-RAY; DRUG DESIGN; HIV-1; HIV-1 REVERSE TRANSCRIPTASE; HUMANS; LIGANDS; MICROBIAL SENSITIVITY TESTS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PYRROLES; REVERSE TRANSCRIPTASE INHIBITORS; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 33846214344 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200600122 Document Type: Article

Times cited : (17)

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