Ortho Functionalization of Aromatic Amines: Ortho Lithiation of N-Pivaloylanilines

Journal of Organic Chemistry

Volumn 44, Issue 7, 1979, Pages 1133-1136

  Fuhrer, Walter ^a   Gschwend, Heinz W ^b  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

^b NOVARTIS PHARMA AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 33845560452     PISSN: 00223263     EISSN: 15206904     Source Type: Journal    
DOI: 10.1021/jo01321a023     Document Type: Article

References (13)

1. Houben-Weyl, “Methoden der Organischen Chemie,” Vol. 11, Georg Thleme Verlag, Stuttgart, 1957, p 1005.
2. G. A. Olah, “Frledel-Crafts and Related Reactions”, Interscience, New York, 1963-1965.
3. P. Claus and W. Vycudlllk, Tetrahedron Lett., 3607 (1968).
4. P. Claus, W. Vycudlllk, and W. Rieden, Monatsh. Chem., 102, 1571 (1971).
5. P. G. Gassman and G. D. Gruetzmacher, J. Am. Chem. Soc., 96, 5487 (1974)
6. T. Sugasawa, T. Toyoda, M. Adachi, and K. Sasakura, J. Am. Chem. Soc., 100, 4842 (1978).
7. M. Walborsky and P. Ronman, J. Org. Chem., 43, 731 (1978).
8. G. L. Mao, I. T. Barnish, and C. R. Hauser, J. Heterocycl. Chem., 6, 475 (1969).
9. W. T. Colwell, K. Yamamoto, P. Christie, and O. W. Henry, Synth. Common., 2, 109 (1972).
10. R. P. Woodbury and M. W. Rathke, J. Org. Chem., 42, 1688 (1977).
11. E. Jung and R. B. Blum, Tetrahedron Lett., 3791 (1977).
12. F. Plozzl and M. R. Langella, Gazz. Chim. Ital., 93, 1382 (1963).
13. Y. Ito, K. Kobayashi, and T. Saegusa, J. Am. Chem. Soc., 99, 3532 (1977).