A Convenient Synthesis of Guanidines from Thioureas

Journal of Organic Chemistry

Volumn 51, Issue 10, 1986, Pages 1882-1884

  Maryanoff, Cynthia A ^a   Stanzione, Robin C ^a   Plampin, James N ^a   Mills, John E ^a  

^a McNeil Pharmaceutical ^*  (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 33845374251     PISSN: 00223263     EISSN: 15206904     Source Type: Journal    
DOI: 10.1021/jo00360a040     Document Type: Article

References (32)

1. Rasmussen, C. R. U.S. Patent 4 211867, 1980.
2. Rasmussen, C. R.; Maryanoff, B. E.; Tutwiler. G. F. Annu. Rep. Med. Chem. 1981, 16, 173.
3. Braun, C. E. J. Am. Chem. Soc. 1933, 55, 1280.
4. King, H.; Tonkin, S. M. J. Chem. Soc. 1946, 1063.
5. McKay, A. F.; Hatton, W. G.; Braun, R.O. J. Am. Chem. Soc. 1956, 78, 6144.
6. Brand, E.; Brand, F. C. “Organic Syntheses”; Wiley: New York, 1955, Collect. Vol. III, p 440.
7. Jen, T.; Van Hoeven, H.; Groves, W.; McLean, R. A.; Loev, B. J. Med. Chem. 1975, 18, 90.
8. “The Organic Chemistry of Drug Synthesis”; Lednicer, D., Mitscher, L. A., Eds.; John Wiley and Sons, Inc.: New York, Vol. I (1977) and Vol. II (1980).
9. Davis, T. L. Org. Synth. 1927, 7, 46.
10. Kampf, A. Chem. Ber. 1904, 37, 1681.
11. Arndt, F.; Rosenau, B. Chem. Ber. 1917, 50, 1260.
12. Rasmussen, C. R. U.S. Patent 4 414 211, 1980.
13. Mikolajczyk, M. M.; Kielbasinski, P. Tetrahedron 1981, 37, 233.
14. Bredereck, H.; Bredereck, K. Chem. Ber. 1961, 94, 2278.
15. Eilingsfeld, H.; Neubauer, G.; Seefelder, M.; Weidinger, H. Chem. Ber. 1964, 97, 1232.
16. Walter, W. Angew. Chem. 1955, 67, 275.
17. Alhede, B.; Gelting, N. C. British Patent 1587258, 1977.
18. Walter, W.; Rohloff, C. Liebigs Ann. Chem. 1975, 295.
19. Pfleiderer, W.; Baur, R.; Bartke, M.; Lutz, H. In “Chemistry and Biology of Pteridines”; Blair, J. A., Ed.; De Gruyter: Berlin 1983; p 93.
20. Walter, W.; Randau, G. Liebigs Ann. Chem. 1969, 722, 98.
21. Walter, W.; Randau, G. Liebigs Ann. Chem. 1969, 722, 80.
22. Hector, D. S. Chem. Ber. 1889, 22, 1176.
23. Hector, D. S. Chem. Ber. 1890, 23, 357.
24. Difuria, F.; Modena, G. Rev. Chem. In. 1985, 6, 51.
25. Sheldon, R. A.; Kochi, J. K. “Metal Catalyzed Oxidations of Organic Compounds’’; Academic Press: New York, 1981.
26. Mimoun, H. “The Chemistry of Functional Groups, Peroxides”; Patai, S., Ed.; John Wiley and Sons: New York, 1982; p 463.
27. Yarovenko, E. Y.; Lastovskii, R. P. J. Org. Chem. USSR (Engl. Transl.) 1970, 6, 952.
28. De Filippo, D.; Ponticelli, G.; Trogu, E. F. J. Chem. Soc., Perkin Trans. 2 1972, 1500.
29. R. K. Harris and B. E. Mann, in “NMR and the Periodic Table”; Academic Press: New York, 1978.
30. Kiselev, L. A.; Shvetsova-Shilovskaya, K. D.; Khanina, L. N.; Mel’nikov, N. N. J. Org. Chem. USSR (Engl. Transl.) 1967, 4, 459.
31. Kiselev, L. A.; Ruchkin, V. E.; Osipova, N. M.; Mel’nikov, N. N.; Shvetsova-Shilovskaya, K. D. J. Org. Chem. USSR (Engl. Transl.) 1966, 2, 2144.
32. Weast, R.C. Ed. “Handbook of Chemistry and Physics”, 51st ed.; CRC Publishing Co.: Cleveland, 1971; 317.