Synthesis and bioactivity of aripiprazole derivatives

Arzneimittel-Forschung/Drug Research

Volumn 56, Issue 10, 2006, Pages 673-677

  Ge, Hai Xia ^a,b   Wang, Li Chen ^a   Jiang, Zhen Zhou ^a   Ni, Sheng Liang ^b  

^a CHINA PHARMACEUTICAL UNIVERSITY   (China)

^b HUZHOU UNIVERSITY   (China)

Author keywords

Antipsychotics, atypical; Aripiprazole, derivatives, dopamine receptor antagonist activity, synthesis; CAS 129722 12 9; Dopamine receptor antagonists

Indexed keywords

1 (5 NITRO 6 AMINO 2 PYRIDINYL)PIPERAZINE; 1 (6 CHLORO 2 PYRIDINYL)PIPERAZINE; 7 HYDROXY 3,4 DIHYDRO 2 (1H) QUINOLINONE; 7 [4 [4 (2 AMINO 4 METHOXY 6 PYRIMIDINYL) 1 PIPERAZINYL]BUTOXY] 3,4 DIHYDRO 2 (1H) QUINOLINONE; 7 [4 [4 (2 AMINO 4 METHYL 6 PYRIMIDINYL) 1 PIPERAZINYL]BUTOXY] 3,4 DIHYDRO 2 (1H) QUINOLINONE; 7 [4 [4 (2,4 DIMETHOXY 6 TRIAZINE) 1 PIPERAZINYL]BUTOXY] 3,4 DIHYDRO 2 (1H) QUINOLINONE; 7 [4 [4 (4 CHLORO 6 PYRIMIDINYL) 1 PIPERAZINYL]BUTOXY] 3,4 DIHYDRO 2 (1H) QUINOLINONE; 7 [4 [4 (4,6 DIMETHOXY 2 PYRIMIDINYL) 1 PIPERAZINYL]BUTOXY] 3,4 DIHYDRO 2 (1H) QUINOLINONE; 7 [4 [4 (6 METHYL 5 NITRO 2 PYRIDINYL) 1 PIPERAZINYL]BUTOXY] 3,4 DIHYDRO 2 (1H) QUINOLINONE; ARIPIPRAZOLE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG EFFECT; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; INFRARED SPECTROSCOPY; MALE; MASS SPECTROMETRY; MOUSE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE;

EID: 33751007307     PISSN: 00044172     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-0031-1296771     Document Type: Article

References (6)

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