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Volumn 41, Issue 9, 2006, Pages 434-441

Sitagliptin: The first dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes

Author keywords

[No Author keywords available]

Indexed keywords

DIPEPTIDYL PEPTIDASE IV; DIPEPTIDYL PEPTIDASE IV INHIBITOR; GLUCAGON LIKE PEPTIDE 1; GLUCOSE; HEMOGLOBIN A1C; INSULIN; METFORMIN; SITAGLIPTIN; UNCLASSIFIED DRUG;

EID: 33749983928     PISSN: 1082801X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review
Times cited : (3)

References (32)
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    • Bergman AJ, Stevens C, Zhou Y, et al. Pharmacokinetic and pharmacodynamic properties of multiple oral doses of sitagliptin, a dipeptidyl peptidase-IV inhibitor: a double-blind, randomized, placebo-controlled study in healthy male volunteers. Clin Ther. 2006;28:55-72.
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    • Abstract PIII-17
    • Krishna R, Bergman AJ, Larson P, et al. Effect of a single cyclosporine A (Neoral) dose on the single-dose pharmacokinetics (PK) of sitagliptin (MK-0431), a dipeptidyl peptidase-IV inhibitor (DPP-IV), in healthy male subjects [abstract]. Clin Pharm Ther. 2006;79;P63. Abstract PIII-17.
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  • 31
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    • Sitagliptin (MK-0431), a selective dipeptidyl-peptidase-IV (DPP-IV) inhibitor, does not affect the pharmacokinetics of simvastatin in humans
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    • Bergman AJ, Cote J, Maes A, et al. Sitagliptin (MK-0431), a selective dipeptidyl-peptidase-IV (DPP-IV) inhibitor, does not affect the pharmacokinetics of simvastatin in humans [abstract]. Clin Pharm Ther. 2006;79;P48. Abstract PII-46.
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    • Bergman, A.J.1    Cote, J.2    Maes, A.3
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    • Bergman AJ, Stevens C, Zhou Y, et al. Pharmacokinetic and pharmacodynamic properties of multiple oral doses of sitagliptin, a dipeptidyl peptidase-IV inhibitor: a double-blind, randomized, placebo-controlled study in healthy male volunteers. Clin Ther. 2006;28:55-72.
    • (2006) Clin Ther , vol.28 , pp. 55-72
    • Bergman, A.J.1    Stevens, C.2    Zhou, Y.3


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