Inhibitors and inactivators of protein arginine deiminase 4: Functional and structural characterization

Biochemistry

Volumn 45, Issue 39, 2006, Pages 11727-11736

  Luo, Yuan ^a   Arita, Kyouhei ^c   Bhatia, Monica ^a   Knuckley, Bryan ^a   Lee, Young Ho ^b   Stallcup, Michael R ^b   Sato, Mamoru ^c   Thompson, Paul R ^a  

^a UNIVERSITY OF SOUTH CAROLINA   (United States)

^b UNIVERSITY OF SOUTHERN CALIFORNIA   (United States)

^c YOKOHAMA CITY UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

BIOCHEMISTRY; CALCIUM COMPOUNDS; CATALYSIS; DISEASES; PHARMACODYNAMICS; PHYSIOLOGY;

CHRONIC AUTOIMMUNE; F-AMIDINE; PROTEIN ARGININE;

PROTEINS;

ARGININE; CALCIUM; CITRULLINE; ENZYME INHIBITOR; N ALPHA BENZOYL N5 (2 CHLORO 1 IMINOETHYL)ORNITHINE AMIDE; N ALPHA BENZOYL N5 (2 FLUORO 1 IMINOETHYL)ORNITHINE AMIDE; ORNITHINE DERIVATIVE; PROTEIN ARGININE DEIMINASE; PROTEIN ARGININE DEIMINASE 4; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CATALYSIS; CATALYST; COMPLEX FORMATION; CONTROLLED STUDY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INACTIVATION; ENZYME INHIBITION; HYDROLYSIS; NONHUMAN; PRIORITY JOURNAL; REACTION ANALYSIS; RHEUMATOID ARTHRITIS; STRUCTURE ANALYSIS; TRANSCRIPTION REGULATION;

AMIDINES; ARGININE; ARTHRITIS, RHEUMATOID; CALCIUM; CHRONIC DISEASE; CITRULLINE; ENZYME ACTIVATION; ENZYME INHIBITORS; HUMANS; HYDROCARBONS, FLUORINATED; HYDROLASES; MOLECULAR PROBES; PROTEIN PROCESSING, POST-TRANSLATIONAL; PROTEIN STRUCTURE, TERTIARY;

EID: 33749359452     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi061180d     Document Type: Article

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