A convenient synthesis of 4-alkyl-5-aminoisoxazoles

Organic Letters

Volumn 8, Issue 17, 2006, Pages 3679-3680

  Bourbeau, Matthew P ^a   Rider, James T ^a  

^a AMGEN INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINE; ISOXAZOLE DERIVATIVE; NITRILE; OXIME;

ALKYLATION; ARTICLE; CATALYSIS; CHEMISTRY; COMBINATORIAL CHEMISTRY; SYNTHESIS;

ALKYLATION; AMINES; CATALYSIS; COMBINATORIAL CHEMISTRY TECHNIQUES; ISOXAZOLES; NITRILES; OXIMES;

EID: 33748605584     PISSN: 15237060     EISSN: None     Source Type: Journal    
DOI: 10.1021/ol061260+     Document Type: Article

References (8)

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7. Presumably, the chloronation occurs during the synthesis of the thienyl (alpha;)-chlorooxime from the corresponding oxime by treatment with n-chlorosuccinimide.
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