Synthesis and structural characteristics of novel 5H-thiazolo[2,3-d][1,5]benzothiazepine derivatives

Journal of the Chemical Society - Perkin Transactions 1

Volumn , Issue 15, 1997, Pages 2211-2215

  Bruno, Giuseppe ^a   Chimirri, Alba ^b   Gitto, Rosaria ^b   Grasso, Silvana ^b   Nicolò, Francesco ^a   Scopelliti, Rosario ^a   Zappalà, Maria ^b  

^a Chim Analitica Chim Fis dell'U   (Italy)

^b Dipartimento Farmaco Chimico   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 33748601623     PISSN: 0300922X     EISSN: None     Source Type: Journal    
DOI: 10.1039/a701539i     Document Type: Article

References (28)

1. A. Chimirri, R. Gitto, S. Grasso, A. M. Monforte and M. Zappalà, Adv. Heterocycl. Chem., 1995, 63, 61.
2. (a) G. Capozzi, A. Chimirri, S. Grasso, G. Romeo and G. Zappia, Heterocycles, 1985, 23, 2051;
3. (b) M. Zappalà, A. Chimirri, S. Grasso, G. Romeo and A. M. Monforte, Il Farmaco, Ed. Sc., 1989, 44, 185;
4. (c) A. Chimirri, S. Grasso, A. M. Monforte, G. Romeo and M. Zappalà, Heterocycles, 1993, 36, 691.
5. A. Chimirri, R. Gitto, S. Grasso, P. Monforte and M. Zappalà, Heterocycles, 1994, 38, 2289.
6. W. Ried and G. Sell, Chem. Ber., 1980, 113, 2314.
7. (a) J. Krapcho, E. R. Spitzmiller and C. F. Turk, J. Med. Chem., 1963, 6, 544;
8. (b) B. Letois, J. C. Lancelot, C. Saturnino, M. Robba and P. De Caprariis, J. Heterocycl. Chem., 1992, 29, 1769.
9. V. Ambrogi, G. Grandolini, L. Perioli, L. Giusti, A. Lucacchini and C. Martini, Il Farmaco, 1993, 48, 665.
10. G. Kaupp and D. Matthies, Chem. Ber., 1987, 120, 1741.
11. D. Cremer and J. A. Pople, J. Am. Chem. Soc., 1975, 97, 1354.
12. M. Nardelli, Acta Crystllogr., Sect. C, 1983, 39, 1141.
13. (a) L. Jiang, S. Liu, G. Li, H. Wu and S. Jin, Chem. Res. Chin. Univ., 1992, 8, 247;
14. (b) L. Jiang, S. Liu, G. Li, H. Wu and S. Jin, Jiegou Huaxue (J. Struct. Chem.), 1992, 11, 297.
15. F. H. Allen, J. E. Davies, J. J. Galloy, O. Johnson, O. Kennard, C. F. Macrae, E. M. Mitchell, G. F. Mitchell, J. M. Smith and D. G. Watson, J. Chem. Info. Comp. Sci. 1991, 31, 187.
16. D. P. Hansell, K. J. Robinson, J. D. Wallis and D. C. Povey, Acta Crystallogr., Sect. C, 1996, 52, 136.
17. The calculations were carried out, on the X-ray refined model, using AMPAC 5.0 program (© 1994 Semichem, 7128 Summit, Shawnee, KS 66216), in which AMI option is included: cf. M. J. S. Dewar, E. G. Zoebisch, E. F. Healy and J. J. P. Stewart, J. Am. Chem. Soc., 1985, 107, 3902.
18. (a) J. G. Angyan, R. A. Poirier, A. Kucsman and I. G. Csizmadia, J. Am. Chem. Soc., 1987, 109, 2237;
19. (b) R. F. Hudson, J. D. Wallis and P. Hansell, Heterocycles, 1994, 37, 1933;
20. (c) A. N. Dixit, K. V. Reddy, A. R. A. S. Deshmukh, S. Rajappa, B. Ganguly and J. Chandrasekhar, Tetrahedron, 1995, 51, 1437;
21. (d) H. Jacobsen, H. K. Kraatz, T. Ziegler and P. M. Boorman, J. Am. Chem. Soc., 1992, 114, 7851.
22. (a) D. H. R. Barton, M. B. Hall, Z. Lin, S. I. Parekh and J. Reibenspies, J. Am. Chem. Soc., 1993, 115, 5056;
23. (b) F. T. Burling and B. M. Goldstein, J. Am. Chem. Soc., 1992, 114, 2313;
24. (c) T. Chivers, I. Krouse, M. Parvez, I. Vargas-Baca, T. Ziegler and P. Zoricak, Inorg. Chem., 1996, 35, 5836.
25. A. Altomare, O. Cascarano, C. Giacovazzo, A. Guagliardi, M. C. Burla, G. Polidori and M. Camalli, J. Appl. Cryst., 1994, 27, 435.
26. G. M. Sheldrick, SHELXTL Plus, Release 4.21, Siemens Analytical X-Ray Instruments Inc., Madison, Wisconsin, USA, 1990.
27. G. M. Sheldrick, SHELXL-93, Program for the Refinement of Crystal Structures, University of Göttingen, Germany, 1993.
28. International Tables for Crystallography, vol. C, ed. A. J. C. Wilson, Kluwer Academic Publishers, Boston, 1992, Tables 4.2.6.8 and 6.1.1.4.