Synthesis of 2,4-disubstituted 5-aminoimidazoles using microwave irradiation

Journal of Combinatorial Chemistry

Volumn 8, Issue 4, 2006, Pages 464-468

  Soh, Chai Hoon ^a   Chui, Wai Keung ^a   Lam, Yulin ^a  

^a NATIONAL UNIVERSITY OF SINGAPORE   (Singapore)

Author keywords

[No Author keywords available]

Indexed keywords

5 AMINOINDAZOLE; 5-AMINOINDAZOLE; INDAZOLE DERIVATIVE;

ARTICLE; CHEMICAL MODEL; CHEMICAL STRUCTURE; COMBINATORIAL CHEMISTRY; MICROWAVE RADIATION; SYNTHESIS;

COMBINATORIAL CHEMISTRY TECHNIQUES; INDAZOLES; MICROWAVES; MODELS, CHEMICAL; MOLECULAR STRUCTURE;

EID: 33746376595     PISSN: 15204766     EISSN: None     Source Type: Journal    
DOI: 10.1021/cc060030j     Document Type: Article

References (25)

1. Shealy, Y. F. J. Pharm. Sci. 1970, 59, 1533-1558.
2. (a) Schrimsher, J. L.; Schendel, F. J.; Stubbe, J.; Smith, J. M. Biochemistry 1986, 25, 4366-4371.
3. (b) Estramareix, B.; David, S. Biochem. Biophys. Res. Commun. 1986, 134, 1136-1141.
4. Cramp, S. M.; Hatton, L. R. Eur. Pat. Appl. EP 283173, 1988.
5. Zhu, Y.; Gross, T. D.; Gao, Y.; Connors, P. J., Jr.; Guo, Z.; Chen, C. PCT Int. Appl. WO 01 29,044. Chem. Abstr. 2001, 134, 311224.
6. Samari, H. R.; Seglen, P. O. J. Biol. Chem. 1998, 273, 23758-23763.
7. (a) Jorgensen, S. B.; Viollet, B.; Andreelli, F.; Frosig, C.; Birk, J. B.; Schjerling, P.; Vaulont, S.; Richter, E. A.; Wojtaszewski, J. F. P. J. Biol. Chem. 2004, 279, 1070-1079.
8. (b) Scott, J. W.; Hawley, S. A.; Green, K. A.; Anis, M.; Stewart, G.; Scullion, G. A.; Norman, D. G.; Hardie, D. G. J. Clin. Invest. 2004, 113, 274-284.
9. (c) Gadalla, A. E.; Pearson, T.; Currie, A. J.; Dale, N.; Hawley, S. A.; Sheehan, M.; Hirst, W.; Michel, A. D.; Randall, A.; Hardie, D. G.; Frenguelli, B. G. J. Neurochem. 2004, 88, 1272-1282.
10. (d) Nath, N.; Giri, S.; Prasad, R.; Salem, M. L.; Singh, A. K.; Singh, I. J. Immunol. 2005, 175, 566-574.
11. (e) Rattan, R.; Giri, S,; Singh, A. K.; Singh, I. J. Biol. Chem. 2005, 280, 39582-39593.
12. (a) Vuilhorgne, M.; Malpart, J.; Mutti, S.; Mignani, S. J. Heterocycl. Chem. 2003, 40, 150-162.
13. (b) Gomez, E.; Avendano, C.; McKillop, A. Tetrahedron 1986, 42, 2625-2634.
14. (c) Rose, C. J.; Rainsworth, A. T. West German Pat., 2 358 509, 1974; Chem. Abstr. 1974, 81, 63630y.
15. (d) Miller, C. S.; Gurin, S.; Wilson, D. W. J. Am. Chem. Soc. 1952, 74, 2892-2894.
16. (e) Bader, H.; Downer, J. D.; Driver, P. J. Chem. Soc. 1950, 2775-2784.
17. (f) Cook, A. H.; Heilbron, I.; Smith, E. J. Chem. Soc. Abstr. 1949, 1440-1442.
18. (a) Yousif, N. M.; Tetrahedron 1989, 45, 4599-4604.
19. (b) Walczynski, K.; Timmerman, H.; Zuiderveld, P. O.; Zhang, M. Q.; Glinka, R. Farmaco 1999, 54, 533-541.
20. (c) Brillon, D. Synth. Commun. 1992, 22, 1397-1401.
21. (d) Benner, S. A. Tetrahedron Lett. 1981, 22, 1851-1854.
22. (a) Baati, R.; Gouverneur, V.; Mioskowski, C. Synthesis 1999, 927-929.
23. (a) Takido, T.; Itabashi, K. Synthesis 1987, 817-819.
24. (b) Walter, W.; Krohn, J. Chem. Ber. 1969, 102, 3786-3794.
25. Logemann, F. I.; Gordon, S. Chem. Ind. 1980, 5, 541-542.