Synthesis and molecular modeling of a lisinopril-tryptophan analogue inhibitor of angiotensin I-converting enzyme

Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 17, 2006, Pages 4616-4619

  Nchinda, Aloysius T ^a   Chibale, Kelly ^a   Redelinghuys, Pierre ^a   Sturrock, Edward D ^a  

^a UNIVERSITY OF CAPE TOWN   (South Africa)

Author keywords

ACE inhibitor; C domain; Hypertension; Molecular docking

Indexed keywords

DIPEPTIDYL CARBOXYPEPTIDASE INHIBITOR; HYDROGEN; LISINOPRIL; TRYPTOPHAN DERIVATIVE;

ARTICLE; DRUG ACTIVITY; DRUG POTENCY; DRUG PROTEIN BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVE SITE; ENZYME INHIBITION; HYDROGEN BOND; HYDROPHOBICITY; MOLECULAR MODEL; PROTEIN DOMAIN;

ANGIOTENSIN-CONVERTING ENZYME INHIBITORS; BINDING SITES; LISINOPRIL; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PEPTIDYL-DIPEPTIDASE A; TRYPTOPHAN;

EID: 33746206287     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2006.06.004     Document Type: Article

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